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2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyridin-2-amine
5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-methyl-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
5-methyl-N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(furan-2-ylmethyl)pyridine-2-carboxamide
3-(2H-1,3-benzodioxol-4-ylmethyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}pyridine
2-(dimethylamino)-2-(2-fluorophenyl)-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}ethan-1-one
N-{[7-(3,3-dimethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
2-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}pyrrolidin-3-yl)benzoic acid
N-(oxan-4-yl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(2-methoxyethyl)[(4-methylphenyl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxamide
2-[1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
3-[ethyl(methyl)amino]-2-methyl-1-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-(methoxymethyl)-5-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidine
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(4-methylpiperazin-1-yl)ethyl]acetamide
N-[1-(4-fluorophenyl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-[({5-[1-(2-amino-2-methylpropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
5-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)-N-ethylpyrimidin-2-amine
N-cyclopropyl-1-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2,6-dimethyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
(4aR,8aS)-1-[2-(3,5-difluorophenyl)acetyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
(1S,5R)-3-(benzenesulfonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-acetamidoacetamide
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-[4-(furan-2-yl)butan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
4-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-chloro-3-fluoro-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
3-({1-[(2-chlorophenyl)carbamoyl]pyrrolidin-3-yl}methyl)benzoic acid
(3S,5S,9S)-5-[(quinolin-6-ylmethyl)amino]-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
N-(2-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[1-(2-phenoxyacetyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-(4-fluoro-3-methylphenyl)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(8-methylquinolin-5-yl)pyridin-4-amine
6-(2-phenoxyphenyl)pyridine-3-carboxamide
9-methoxy-4-[(4-methylphenyl)methyl]-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-2-yl}pyridine
N-butyl-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-(3-methoxypropyl)-1-(4-methyl-1,3-thiazol-2-yl)piperidine
3-[1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)pyrrolidin-2-yl]pyridine
N-(butan-2-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-hydroxy-1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-chloro-3-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-pyrazol-5-amine