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ethyl 1-[(4-methoxyphenyl)methyl]-5-(1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(azocan-1-yl)-3-[5-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-cyclopropyl-2-ethyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}butanamide
N-(2-methyl-1-{7-[2-(pyridin-4-ylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
methyl[(5-methylfuran-2-yl)methyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
6-[(1-ethyl-1H-pyrazol-3-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-({7-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
N-cyclopropyl-3-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}propanamide
1-cyclobutanecarbonyl-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-({8-[2-(thiophen-2-yl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
N-cyclopropyl-N-(1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
2-(2-fluorophenyl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-amino-6-[4-(piperidin-1-yl)phenyl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
N-(2-methoxyethyl)-4-methyl-3-{[(2-methylpropyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-(5-acetylpyridin-2-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[6-(4-methoxy-3-methylphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
(1S,2S)-2-(4-{3-azaspiro[5.5]undecan-9-yl}piperazin-1-yl)cyclohexan-1-ol
1-[3-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
2-[3-(2-ethylphenyl)phenyl]ethan-1-amine
2-methyl-4-{5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}but-3-yn-2-ol
(3S,4R)-1-[3-(3,5-dimethylphenyl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
N-cyclopropyl-3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-3-yl}propanamide
7-(2-hydroxyethyl)-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
6-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-[2-(3-chlorophenyl)ethyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-amino-N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N5-[(1-cyclopentylpiperidin-4-yl)methyl]-N6-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
6-methyl-1-[3-oxo-3-(thiomorpholin-4-yl)propyl]-1,2-dihydropyridin-2-one
N,N-dimethyl-4-{4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]piperidin-1-yl}benzamide
N-(3-sulfamoylphenyl)-4-(thian-4-yl)piperazine-1-carboxamide
N-(1-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)methanesulfonamide
3-ethyl-1,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,2-dimethylpropyl)-3-hydroxy-3-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(5-fluoro-2-methylphenyl)methyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-[3-(3,4-dimethylphenyl)propanoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-{4-[2-(4-hydroxyphenyl)-1H-imidazol-1-yl]phenyl}pyridine-3-carboxamide
(1S,5R)-3-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
1-[3-(3-aminoazepan-1-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
N-ethyl-5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyrimidin-2-amine
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-[4-(methylsulfanyl)phenyl]acetamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-6-ol
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methyl-N-(2-methylprop-2-en-1-yl)acetamide
4-(cyclopropylmethyl)-1-[2-(2,3,4-trifluorophenyl)acetyl]-1,4-diazepan-5-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 2-{2-[(2-acetamidoacetamido)methyl]-5-methyl-2,3-dihydro-1-benzofuran-7-yl}benzoate
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]pyrrolidine-2-carboxamide
5-[(8-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine