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1-{3-[(2-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-N,N-diethylpiperidine-3-carboxamide
{1-[1-(6-ethyl-4-methylquinolin-2-yl)piperidin-4-yl]piperidin-3-yl}methanol
2-(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
methyl 2-{3-methyl-4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-oxopiperazin-1-yl}acetate
2-(3-methylbenzamido)-7-oxo-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-({methyl[1-(pyridin-2-yl)propyl]amino}methyl)benzamide
3-({2-[1-(benzenesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{1-[3-(4-fluorophenyl)-3-phenylpropanoyl]piperidin-4-yl}acetamide
1-(2,3-dimethylphenyl)-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-4-amine
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyridine
N,N-dimethyl-5-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
1-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-2-yl)methyl]pyrrolidine
(1S,6R)-9-{[5-(pyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
{[3-({1-[3-(4-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(1,3-thiazol-4-ylmethyl)amine
(2E)-1-[(4aR,8aS)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(3-fluorophenyl)prop-2-en-1-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
5-cyclopropyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-oxazole-4-carboxamide
N-{2-[2-(4-chlorophenoxymethyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}acetamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbutanamide
7-hydroxy-6-methyl-4-(piperidin-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
8-fluoro-N-methyl-N-(oxan-2-ylmethyl)quinoline-2-carboxamide
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-6-methylpyridine-3-carboxamide
2-{[4-(5-chlorothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
1-tert-butyl-N-[3-(2-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
methyl(1,2-oxazol-3-ylmethyl)[(3-{[1-(3,4,5-trimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl]amine
N-cyclopropyl-N-(naphthalen-1-ylmethyl)oxolane-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
ethyl 2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
N-[(2R,3R)-1'-(2-hydroxy-5-methoxybenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-[2-(3-methoxyphenyl)acetyl]piperazin-2-one
2-(4-methylpiperidin-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
N-(2-methoxyphenyl)-2-[4-(4-methylpiperazine-1-carbonyl)morpholin-3-yl]acetamide
1-[1-(3-methylbutanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-(2-ethoxyphenyl)-1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazole
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}amino)-2-methyl-N-(2-methylpropyl)benzamide
[(1R)-1-(4-methoxyphenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[4-(5-chlorothiophen-2-yl)phenyl]-N-methylacetamide
N'-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}ethanediamide
3-(4-fluorophenyl)-4-[3-(methylsulfanyl)propanoyl]piperazin-2-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-(3-methylbutyl)-1H-pyrazole-4-carboxamide
1-[(4-{[1-(2,4-difluorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(2-fluorophenyl)piperazine
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazole
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[2-(pyridin-3-yloxy)ethyl]-1H-1,3-benzodiazole-7-carboxamide
8-(2-acetylbenzoyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,1-dimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)propyl]urea