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{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}(thiophen-3-ylmethyl)amine
1-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
[(3R,4R)-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-methyl-4-(4-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)but-3-yn-2-ol
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(5S,9aS,9bS)-2-cyclopentyl-5-(2,4,5-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azocane
methyl (2S,4R)-4-(dimethylamino)-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxylate
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-methoxypyridin-4-ol
N-(furan-3-ylmethyl)-4-(pyrrolidine-1-sulfonyl)benzamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,4-dithiepan-6-amine
7-(5-chloropyridin-2-yl)-4-(3,5-dimethoxybenzoyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopentyl-4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 4-({[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)-3-methylbenzoate
4-{1-[1-(2,2-dimethylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
N-(furan-2-ylmethyl)-4-{[(6-hydroxypyrimidin-4-yl)methyl]amino}pyridine-2-carboxamide
2-(3-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
4-[(diethylamino)methyl]-5-ethyl-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)furan-2-carboxamide
2-(2,4-dimethoxyphenyl)-8-methoxy-5-(quinolin-7-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-[1-(pyrrolidine-1-carbonyl)azepan-3-yl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
N-(2,3-dihydro-1H-inden-5-yl)-4-(2-phenoxyacetyl)piperazine-1-carboxamide
3-benzyl-4-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperazin-2-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
3-(2-chlorobenzoyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-methoxy-N-(2-methoxyethyl)-2-{[1-(quinolin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
7-[(4-fluorophenyl)methyl]-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenoxypropanamide
N-{1-[7-(2,4-difluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
N-[1-(2,5-dimethylphenyl)ethyl]-2-{2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
[7-(1H-imidazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(2-{[1-(pyridin-2-yl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
5-(3-phenylpropyl)-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[1-(2-phenylethyl)-5-[1-(propan-2-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-chloro-3-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
4-(2,3,6-trimethylquinoline-4-amido)oxane-4-carboxylic acid
3-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-9-methyl-3,9-diazaspiro[5.6]dodecane
N-(3-chloro-4-fluorophenyl)-3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]propanamide
N-[(2-ethoxypyridin-3-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
5-(morpholin-4-yl)-2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(2,3-dihydro-1H-inden-5-yl)propanamide
2-(4-{[3-(morpholin-4-yl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
1-methyl-5-(4-methylpiperazin-1-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide