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N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
N-ethyl-2-(4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
3-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]pyrimidin-2-amine
5-(furan-3-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
dimethyl({2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-1-(3-methylthiophen-2-yl)ethyl})amine
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidine-3-carbonyl)pyridine
methyl 3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
1-[(4-methoxyphenyl)methyl]-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-2-one
methyl 5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 1-benzyl-5-(benzylamino)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
6-fluoro-2-({[(1-propyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-4-ol
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]thiophene-2-sulfonamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-1-(pyridine-4-carbonyl)piperidin-4-amine
4-({[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
2-{[5-cyclopropyl-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-methoxy-4-(3-methyl-1H-pyrazol-1-yl)phenyl]acetamide
methyl (2S)-1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-yl]pyrrolidine-2-carboxylate
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclohexyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
(3S)-3-ethyl-4-{[3-(furan-2-yl)phenyl]methyl}morpholine
4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-methylpiperazin-2-one
8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5,5-diphenyl-1-[2-(pyrazin-2-yl)ethyl]piperidin-2-one
2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}pyrimidine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-benzyl-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(5-fluoro-1,3-dimethyl-1H-indol-2-yl)formamido]acetic acid
1-(2-aminoethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
8-{5-methylthieno[2,3-d]pyrimidin-4-yl}quinoline
N-ethyl-5-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)pyrimidin-2-amine
7-[(2,3-difluorophenyl)methyl]-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N1-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-N4-(furan-2-ylmethyl)piperidine-1,4-dicarboxamide
N-methyl-N-{2-phenyl-1-[1-(3-phenylpropyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-(cyclohexylmethyl)-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1R,5R)-3-methanesulfonyl-6-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]benzonitrile
4-(4-methoxy-3,5-dimethylphenyl)thiophene-2-carboxamide
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(2-methoxyphenyl)-2-methylpiperazine
2-methoxy-4-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]pyridine-3-carbonitrile
1-[4-(3-acetylphenyl)phenyl]-3-[2-(propane-2-sulfonyl)ethyl]urea
5-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,2,3,4-tetrazole
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide