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8-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
dimethyl[2-({1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}oxy)ethyl]amine
(2S,4S)-4-amino-N-ethyl-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
(3S,9aR)-8-(2-methoxybenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
(1R,2S,9R)-11-[2-(2,3-difluorophenyl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(3-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(pyridin-3-yl)ethyl]urea
N-{2-[2-(pyridin-2-ylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
4-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
4-({4-methyl-5-[1-(2-methylpropyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
(1S,5R)-3-(3,6-dimethyl-1-benzofuran-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(6-phenoxypyridin-3-yl)-1-(3-phenylpropyl)piperidine-4-carboxamide
(4aS,7aR)-1-(4-methyl-2-oxopentanoyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-(5-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}thiophen-2-yl)acetamide
4-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-2,6-dimethylphenol
3-({3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1H-indole
N-[(2,3-dimethoxyphenyl)methyl]-3-propanamidobenzamide
N-[(1-methylpiperidin-4-yl)methyl]-3-phenoxy-N-(2-phenylethyl)propanamide
2-[4-({[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
N-(2-oxooxolan-3-yl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(3-fluoropyridine-4-carbonyl)piperidin-3-yl]propanamide
ethyl 4-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}-3,5-dimethyl-1H-pyrrole-2-carboxylate
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(3-methylpyridin-2-yl)methyl]benzamide
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4,6-dimethylpyridine-3-carbonitrile
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 4-benzyl-1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)piperidine-4-carboxylate
2-(2-ethyl-1H-imidazol-1-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2,2-dimethylpropan-1-one
N5-{[2-(difluoromethoxy)phenyl]methyl}-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
1-(azepan-1-yl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
3-(but-2-yn-1-yl)-5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(2S)-2-{2-[(2-ethoxyphenyl)carbamoyl]acetamido}-3-(1H-indol-3-yl)propanoic acid
2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-N-(2-fluoro-4-methylphenyl)acetamide
N3-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)piperidine-1,3-dicarboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(1-phenylcyclopentyl)methyl]pyrimidin-2-amine
N-cyclopentyl-1-ethyl-N-[(4-methylphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-ethyl-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
4-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]pyridine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-ethyl-6-oxopiperidine-3-carboxamide
{1-[1-(3-cyclopentylpropyl)piperidin-3-yl]piperidin-4-yl}methanol
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(thiophen-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(2-fluorophenyl)methyl]-N-(2-methoxy-2-methylpropyl)-6-oxopiperidine-3-carboxamide
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyridine-4-carboxamide
1-(4-methoxyphenyl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclopentane-1-carboxamide
10-methoxy-5-(pyridin-4-ylmethyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2,4-dimethyl-N-(2-{7-[(2E)-4-methylpent-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-(6-cyanopyridin-3-yl)-3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)benzamide
N-ethyl-N-(2-hydroxyethyl)-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide