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N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-methylphenyl (7R,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(propan-2-yl)-1-[(1s,4s)-4-{[(2,3,4-trimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-1-(4-fluoro-2-methylbenzoyl)-4-propylpyrrolidin-3-amine
N-benzyl-N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl 1-(2-methoxyethoxy)-8-(naphthalene-1-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-yl)piperidin-4-ol
3-(azepane-1-carbonyl)-N-[(3-methoxyphenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
4-[2-(benzyloxy)acetyl]-1,3-dimethylpiperazin-2-one
1-(3-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(quinoline-6-carbonyl)pyrrolidin-3-amine
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-(dicyclopropylmethyl)-N-methylacetamide
2-[(3-chlorophenyl)methyl]-4-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclobutylpiperidine-4-carboxamide
(1R,3S)-7-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-methoxy-7-azaspiro[3.5]nonan-1-ol
methyl 3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(5S)-5-{[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyridin-2-ylmethyl)amino]methyl}pyrrolidin-2-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
N-[(2,4-dichlorophenyl)methyl]-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(1-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[(1-methylpiperidin-3-yl)methyl]benzamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}piperidine-3-carboxamide
4-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-chlorophenyl)urea
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-3-methylpyridine-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1H-imidazol-1-yl)ethyl]piperidine-3-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1H-1,2,4-triazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(5-methylthiophen-2-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
6-ethyl-1,5-dimethyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-dihydropyridin-2-one
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazole
1,9-dimethyl-4-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-ethyl-N-(furan-2-ylmethyl)-7-(2-methoxybenzamido)-1-methyl-N-(prop-2-yn-1-yl)-1H-1,3-benzodiazole-5-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
5-methanesulfonyl-2-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyrimidin-4-amine
N-[2-(4-{[2-(4-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-methylphenoxy)ethan-1-one
N-(3-hydroxypropyl)-5-methyl-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
4-({2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[3-(pyrimidin-5-yl)phenyl]acetamide
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-4-methoxy-3,5-dimethylpyridine
5-ethyl-2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
5-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}propanamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
N-[2-(3-acetamidophenyl)phenyl]-2-methoxyacetamide