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methyl 3-[(3-ethoxyphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
7-methyl-3-(2-methylpropyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2-chloro-4-fluorophenyl)-1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
(3R,4R)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
2-cyclopentyl-9-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(furan-3-ylmethyl)-3-(2-oxo-2-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethyl)piperazin-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-methylpropyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
methyl N-(2-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)carbamate
N-cyclopentyl-N-({4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-fluorophenyl)ethyl]propanamide
N-[3-(3-methoxyphenyl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
[1-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
N-cyclopropyl-5-(dimethyl-1,2-oxazole-4-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-chlorophenyl)-5-methyl-4-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]piperazin-2-one
2-chloro-4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}phenol
3-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}propanamide
1-ethyl-3-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-cycloheptyl-3-methoxybenzamide
1-cyclobutanecarbonyl-4-[4-(1H-imidazol-1-yl)benzoyl]-1,4-diazepane
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
9-(2-methanesulfonylacetyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,2,2-trifluoroethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
methyl (2S,3S)-3-methyl-2-({5-[(quinolin-6-yloxy)methyl]-1,2-oxazol-3-yl}formamido)pentanoate
1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-methyl-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
4,6-dimethyl-3-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2S)-2-[3-methyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1-phenylpropan-2-amine
4-benzoyl-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
N-[(2R,3R)-2-ethoxy-1'-propanoyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
ethyl 1-(prop-2-en-1-yl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
[1-(5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
2-(2-chloro-4-fluorophenyl)-N-[(1,4-dimethylpiperazin-2-yl)methyl]acetamide
methyl (1R,3S,3aR,6aS)-1-(2-methoxy-2-oxoethyl)-5-methyl-3-(2-methylphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-cyclopropyl-1-{1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
7-fluoro-4-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)quinolin-2-amine
2-(dimethylamino)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methylphenyl)acetamide
N-(2-fluorophenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
1-(pyrrolidin-3-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperazine
6-(cyclopropylmethoxy)-4-(1-phenylcyclopropanecarbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-(4-methoxyphenyl)-1-[(pyrimidin-4-yl)amino]propan-2-ol