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1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide
{3-[1,5-dimethyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]phenyl}methanol
4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-cycloheptyl-4-[(1-propylpiperidin-4-yl)amino]pyrrolidin-2-one
6-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
1-methyl-4-{1-[1-(pyridine-4-carbonyl)piperidin-4-yl]ethyl}piperazine
2-[2-(dimethylamino)ethyl]-9-(4-ethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-5-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-(4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)acetamide
4-fluoro-3-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]benzene-1-sulfonamide
2-(3,4-dimethoxyphenyl)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-[1-(cyclopropylmethyl)-4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidin-4-amine
N-benzyl[(2H-1,3-benzodioxol-5-yl)amino]sulfonamide
N-(1-hydroxybutan-2-yl)-3-(2-methylpropanamido)-N-(thiophen-2-ylmethyl)benzamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
4-{[3-(2-methyl-1H-imidazol-4-yl)phenyl]methyl}morpholine
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3-benzyl-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
4-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H-imidazol-2-yl)pyridine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(2-{[(cyclopropylmethyl)(methyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
2-methyl-N-(2-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
3-(4-fluoro-3-methylphenyl)-6-(2-phenoxyacetyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
2-methyl-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
5-(2,6-dimethoxyphenyl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,2,4-triazin-3-amine
N-(2,3-dihydro-1H-inden-2-yl)-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]acetamide
N-[(3-chlorophenyl)methyl]-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(diethylamino)-3-[2-methoxy-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
8-(oxan-3-yl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-{2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
2-[(3-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
methyl 3-[(2-chloro-4-fluorophenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1-methyl-1H-indazole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
4-benzyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1H-indazole-3-carboxamide
3-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
4-(dimethylamino)-N-(2-phenoxyphenyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
1-{5-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one