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N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidin-3-yl]cyclopropanecarboxamide
6-methoxy-N-methyl-N-(quinoxalin-2-ylmethyl)pyrimidin-4-amine
1-(azepan-1-yl)-3-[3-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]propan-2-ol
(2E)-1-[(4aR,8aS)-6-[2-(4-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-methylbut-2-en-1-one
3-[4-(dimethylcarbamoyl)phenyl]-4-methylbenzamide
methyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
ethyl 4-(3-{[(adamantan-1-yl)amino]methyl}-6-methylquinolin-2-yl)piperazine-1-carboxylate
3-[(4-fluorophenyl)methyl]-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,2-oxazole-5-carboxamide
1-(azepan-1-yl)-3-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}piperidine-4-carboxamide
N-methyl-N-(2-phenylethyl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-amine
N-(2-methylprop-2-en-1-yl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
4-[3-(3-fluorophenyl)benzoyl]piperazine-1-sulfonamide
7-chloro-2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1-methyl-1H-indole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(oxan-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,9S)-11-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
2-(4-{4-[(butan-2-yl)amino]piperidin-1-yl}phenyl)-1-(pyrrolidin-1-yl)ethan-1-one
4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-methoxypyridine-3-carbonitrile
3-{5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
9-(2-aminopyrimidin-4-yl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-2-(dimethylamino)-N-methylacetamide
1-[(3-methylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazine
5-(2H-1,3-benzodioxol-5-yl)-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,2,4-triazin-3-amine
1-cyclohexyl-N-methyl-N-(quinolin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-(azetidine-1-carbonyl)-5-(cyclobutylmethoxy)benzoate
1-[4-(dimethylamino)azepan-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
N-[(1-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-4-yl)methyl]acetamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-fluorobenzene-1-sulfonamide
N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl){[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
2-ethyl-9-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
methyl 5-[(2-methylpropyl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[1-(2-methylbenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-(oxolane-2-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,6-dioxo-N-propyl-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
4-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidine
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
(5-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
methyl 3-(5-methylpyrazine-2-carbonyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-(1H-indol-3-yl)acetamide