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3-[(2,6-dimethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-1-oxa-8-azaspiro[4.5]decane
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-5-propyl-1,2-oxazole-3-carboxamide
(2R,6R)-1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-(4-fluorophenyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1,4-diazepane
1-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yloxy)ethan-1-one
3,4-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-methanesulfonylpiperidine
1-(3-fluorophenyl)-3-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-({4-[1-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)-1H-1,2,3,4-tetrazole
3-(methanesulfonylmethyl)-1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidine
methyl 4-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]-4-oxobutanoate
ethyl 4-(oxan-2-ylmethyl)-1-(3-phenylprop-2-ynoyl)piperidine-4-carboxylate
2-methoxy-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
N-cyclopropyl-3-{5-[2-(methylsulfanyl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-amino-N-[1-(4-methoxyphenyl)propyl]-N-methylpyridine-4-carboxamide
1-cyclopentyl-4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperazin-2-one
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclobutan-1-amine
3-methyl-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
4-{5-[(methylsulfanyl)methyl]-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
3-[({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-6-ethyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}-3-methylthiophene-2-carboxamide
(1-methyl-5-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-methoxy-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
3-(5-oxo-1-propylpyrrolidin-3-yl)-1-(quinolin-5-yl)urea
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
(3S,4S)-4-cyclopropyl-1-[(2-phenylethyl)carbamoyl]pyrrolidine-3-carboxylic acid
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
methyl 1-benzyl-5-(cyclopentylamino)-3-cyclopropaneamido-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4R)-4-amino-N-methyl-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidine-2-carboxamide
4-(2-methylphenoxy)-1-[3-(pyrrolidin-3-yl)benzoyl]piperidine
methyl 1-(benzyloxy)-2-oxo-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[1-(2-acetamidoacetyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyrazine-2-carboxamide
1-(4-{[(1-benzothiophen-2-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(2-methylpropyl)acetamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
(2S,4S)-4-(4-{4-[(4-hydroxypiperidin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(5-methylfuran-2-yl)methyl](oxolan-2-ylmethyl)amine
2-(2H-1,3-benzodioxol-5-yl)-5-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-[4-(4-acetylpiperazine-1-carbonyl)piperidin-1-yl]-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-4-carboxamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
8-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[4-(1-ethyl-5-oxopyrrolidine-3-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
2-ethyl-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)butanamide