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N-[2-(2-chlorophenyl)ethyl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-(azocane-1-carbonyl)-N-(propan-2-yl)pyrimidin-2-amine
2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1-methyl-1H-1,3-benzodiazole
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-cyclopropylpiperidin-2-one
N-cyclopropyl-1-(2-{1-[(2-methoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
1-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1,5-dimethyl-2-phenyl-4-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
8-[(4-hydroxy-3-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-3-methoxy-N-(pyridin-3-ylmethyl)benzamide
1-(propan-2-yl)-4-[4-(3,4,5-trimethoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
(3S,4R)-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-({8-[(3,4-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,3-thiazole-5-carboxamide
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylquinolin-8-yl)urea
2-methyl-4-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-1,4-oxazepane
5-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[3-(oxolan-3-yl)propyl]-1-[3-(trifluoromethoxy)phenyl]urea
2-(cyclopropylmethyl)-8-[3-(2-fluorophenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(diethylamino)ethyl]-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
2-[(2-benzylmorpholin-4-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
(1S,5R)-3-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-acetyl-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]thiophene-2-carboxamide
{2-oxo-2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}urea
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-cyclopropyl-1-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
3-{5-[3-(4-hydroxyphenyl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-(5-amino-1-methyl-1H-pyrazol-4-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
4-benzoyl-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(3-methoxybenzoyl)piperazine
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-cyclopentyl-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-methyl-1-[4-(naphthalene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
2-({4-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
3-methyl-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
(2S,4S)-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
methyl 8-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
7-(3-chlorophenyl)-4-(1,3-thiazole-5-carbonyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridine
5-[(3,4-dimethoxyphenyl)methyl]-5-{3-[4-(2,3-dimethylphenyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
8-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(adamantan-1-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
5-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-1,2,3-benzotriazole
5-(1-benzoylpiperidin-4-yl)-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(3,4-dimethoxyphenyl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide