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N-(1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methoxybenzoyl)-4-[(2R)-pyrrolidine-2-carbonyl]piperazine
methyl 3-{2-[4-(methylsulfanyl)phenyl]acetyl}-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
dimethyl({5-[1-(6-methylpyridin-3-yl)-1H-imidazol-2-yl]thiophen-3-yl}methyl)amine
4-{1-ethyl-5-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-3-yl}pyridine
4-[2-(2-methoxyphenoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(thiophen-3-ylmethyl)piperidine
1-{6-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyridin-3-yl}ethan-1-one
5-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidine-1-carbonyl)-1,3-benzothiazol-2-amine
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(2R)-3-(benzyloxy)-2-[5-(1-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
(1r,4r)-4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[(4-phenylphenyl)methyl]amine
5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-2-methoxybenzamide
2,3,5-trimethyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-[1-(2-hydroxyethyl)-3-[(1-phenylethyl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
2-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[(1-propyl-1H-imidazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}acetamide
4-[(2-amino-5-methylpyrimidin-4-yl)amino]-1-(4-chlorophenyl)pyrrolidin-2-one
N-(1-{7-[2-(2-chlorophenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(pyrrolidin-1-yl)acetamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
3-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-[(3,4-difluorophenyl)methyl]-8-[(2S)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-(2,4-dichlorophenyl)-5-(morpholin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
6-methyl-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
2-({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})amino)ethan-1-ol
N-(pyridin-4-ylmethyl)-4-{[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-{3-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]propyl}pyrrolidin-2-one
2-benzyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,3-benzoxazole-5-carboxamide
[(4-methanesulfonylphenyl)methyl](methyl)[1-(pyridin-3-yl)propyl]amine
1-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-oxoethyl}-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-benzyl-1-(3-methoxypropyl)-8-[3-(methylsulfanyl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
2-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
5-methyl-3-{2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[1-(cyclopentylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-({3-methyl-7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
2-(3-chloro-4-hydroxyphenyl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
8-cyclopentyl-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-(2-hydroxyethyl)-4-(quinoxaline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-ethyl-4-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)-3-methylpiperazin-2-one
9-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(2-methyl-1,3-benzoxazole-6-carbonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
4-chloro-1-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
(3S,7S,8aS)-7-{[(2,5-difluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione