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4-(1-methylpiperidin-4-yl)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
1-cyclobutanecarbonyl-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
3-(4-hydroxyphenyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-methyl-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]pyrrolidine-3-carboxamide
5-cyclopropyl-N-(3-ethoxypropyl)-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-(piperidin-3-yl)pyrimidin-4-amine
2-{4-[1-(2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxylate
7-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
1-(2-ethoxyphenyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
(1R,2S,6R,7S)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-4-oxobutane-1-sulfonamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-ethenylpyridine
9-ethyl-4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 3-benzyl-1-[(2-methoxyphenyl)carbamoyl]piperidine-3-carboxylate
N,N-diethyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-5-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)pyrimidin-2-amine
1-[2-(4-methanesulfonyl-1,4-diazepan-1-yl)pyrimidin-4-yl]piperidin-3-ol
6-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-1,6-dihydropyridine-3-carboxamide
2-(methylsulfanyl)-N-[2-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
3-[1-(2,6-dimethylquinoline-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
4-ethyl-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-fluoro-N-[3-(furan-2-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
methyl 3-(3-fluorobenzamido)-6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
4-[(1S,2S)-2-hydroxycyclohexyl]-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperazine-1-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(propan-2-yl)benzamide
N-{[3-methyl-7-(2-phenoxyacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
5-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
3-[({2-[(dimethylamino)methyl]phenyl}methyl)amino]pyrazine-2-carbonitrile
(3R,9aR)-8-[(4-chlorophenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
8-chloro-4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-2-methylquinoline
5-{[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-amine
8-methoxy-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(isoquinolin-5-ylmethyl)-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(oxolan-3-yl)-3-{[3-(1H-1,2,4-triazol-1-yl)propyl]sulfamoyl}benzamide
4-benzyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}propan-1-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
2-({4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-4,6-dimethylpyrimidine
1-(5-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-2-methylphenyl)imidazolidin-2-one