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(3aR,6aR)-2-methyl-N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
[1-(4-methylphenyl)propan-2-yl][1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]amine
2-phenyl-N-[2-(pyridin-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N,3,6-trimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1-benzofuran-2-carboxamide
(2R,6R)-4-(3-propyl-1H-pyrazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1,4-dihydroquinolin-4-one
N-(2-fluorophenyl)-3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
5'-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]
methyl 2-{[(2-methylbutan-2-yl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
8-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(4-fluorophenyl)-2,2-dimethyl-N-[3-(methylsulfanyl)propyl]cyclopropane-1-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
4-{[1-(3-cyclopentylpropyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
methyl 3-{[(2,3-dimethyl-1H-indol-7-yl)formamido]methyl}-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
3-(3-methoxyphenyl)-N-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazole
5-[1-(4-chlorophenyl)cyclobutyl]-1-methyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
4-(2-methoxyphenyl)-2-methyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
2-(4-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(2-aminoethyl)-N-[2-(dimethylamino)ethyl]-N-[(4-methylphenyl)methyl]quinazolin-4-amine
(1S,5R)-3-(1H-1,2,3-benzotriazole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-3-[(5-chlorothiophen-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}quinoline
{2-[(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)methyl]phenyl}methanol
N-(1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
7-fluoro-3-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)-1,2-dihydroquinolin-2-one
4-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-[(3-fluorophenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-phenyl-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
2-ethoxy-N-ethyl-N-[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]pyridine-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-{3-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}propan-2-ol
3-[(3R,4S)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
3,5-dimethyl-2-{[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}pyridin-4-ol
4,4,4-trifluoro-1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-6-(piperidine-1-carbonyl)pyrazine
8-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({[(4-ethylphenyl)methyl](2-methoxyethyl)amino}methyl)-6-fluoroquinolin-4-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
2-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}quinolin-4-ol
(3aR,6aS)-2-ethyl-5-{[(3-fluorophenyl)methyl]carbamoyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-{2-[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
8-(4-chloro-1-methyl-1H-indole-2-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one