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2,3,5,6-tetramethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methoxypyridine
3-butyl-4-(5-hydroxypyrazine-2-carbonyl)-1-methylpiperazin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3R,4S)-4-(4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)oxolan-3-ol
2-{2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenoxy}ethan-1-ol
N-(3-cyanophenyl)-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
5-fluoro-2-(1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-(2,3-dihydro-1H-inden-1-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
4-(1-methyl-1H-imidazol-2-yl)-1-[2-(oxolan-3-yl)ethyl]piperidine
1-(2-methoxyethyl)-3-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid
(3R,5S)-5-(3-fluorophenoxymethyl)-1-(naphthalen-2-ylmethyl)-N-(2-phenylethyl)piperidine-3-carboxamide
1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
7-methyl-3-{[2-(5-methylfuran-2-yl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
N-(pyridin-3-ylmethyl)-4-(quinoxalin-2-yl)piperazine-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(oxolan-2-ylmethyl)acetamide
2-(3-fluorophenyl)-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidine
(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenoxyethyl)acetamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-cyclopropyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)morpholine
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4-phenyl-1,4-diazepane
4-{2-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethoxy}-3-methoxybenzoic acid
2-(dimethyl-1,3-thiazol-5-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
2-(4-hydroxyphenyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-cyclopropyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[1-({1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-methoxypyridine-4-carboxamide
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol
N-cyclohexyl-N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
5-ethyl-2-methyl-4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-[4-(3-fluorophenyl)phenyl]-N-[3-(methylamino)propyl]piperidin-4-amine
(3E)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]hex-3-en-1-one
2-{5-[(2,5-dioxoimidazolidin-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
8-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-3-ol
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-cyclopentylpiperazine
2-(2H-1,3-benzodioxol-5-yl)-3-methylquinoxaline
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(1R,5S)-6-[(3,5-dichloropyridin-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
9-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-3-oxa-9-azaspiro[5.5]undecane
7-(3-chlorophenyl)-4-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]morpholine