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(2S,4S)-4-amino-N,N-diethyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidine-2-carboxamide
(3aS,6aS)-2-benzyl-5-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-chloro-6-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxylic acid
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-[3-(pyridin-4-yl)propyl]acetamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
1-[2-(4-chlorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-(3-methylbutyl)-2-oxo-3-(pyridin-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
(1S,5R)-N-(3-cyanophenyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(4aS,8aR)-6-(2,3-dimethoxybenzoyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-(methoxymethyl)-5-(oxolan-2-ylmethyl)-1,3-benzoxazole
4-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidin-4-yl}pyridine
{5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
N-(furan-2-ylmethyl)-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-(prop-2-yn-1-yl)propanamide
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
(2S)-2-amino-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
N-benzyl-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidine-4-carboxamide
N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)pyrimidine-5-carboxamide
N-[2-(2-fluorophenyl)ethyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2-(4-chloro-2-methylphenoxy)-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]acetamide
7-(cyclopropylmethyl)-2-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
7-[1-(methoxymethyl)cyclobutanecarbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(furan-3-ylmethyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(4aS,8aR)-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)-decahydroisoquinoline
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
1-(cyclohexylmethyl)-N-methyl-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
2-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]furan-2-yl}-1-methyl-1H-1,3-benzodiazole
4-({1-[2-(4-fluorophenoxy)ethyl]piperidin-2-yl}methyl)morpholine
5-{5-[2-(2-fluorophenyl)phenyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
ethyl (4aR,6R,8aS)-2-(1-methyl-1H-pyrazole-3-carbonyl)-6-(morpholin-4-yl)-decahydroisoquinoline-8a-carboxylate
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1H-imidazol-2-ylmethyl)(methyl)[2-(2-methylpiperidin-1-yl)ethyl]amine
3-(2-fluorophenyl)-6-[5-(methoxymethyl)thiophene-2-carbonyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[3-(3,4-diethoxyphenyl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(4-methoxyphenyl)methyl]-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-(3-methoxypropanamido)-N,1-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
(1H-imidazol-2-ylmethyl)(methyl)[2-(4-methylphenoxy)ethyl]amine
2-(2-{[ethyl(pentan-2-yl)amino]methyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
4-fluoro-2-[4-(piperidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]phenol
3-fluoro-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]benzonitrile
(1R,7S)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3R,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-ethyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-methyl-1H-pyrazole-4-carboxamide