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{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}urea
2-({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(4-methoxy-3-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[(4-methyl-1H-imidazol-5-yl)methyl]-8-azabicyclo[3.2.1]octane
8-[3-(2-oxopyrrolidin-1-yl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(2-aminoacetyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(3aR,6aS)-2-[5-(methoxymethyl)furan-2-carbonyl]-octahydropyrrolo[3,4-c]pyrrole
(1S,5R)-3-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-ethoxyphenyl)ethan-1-one
1-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperidine-4-carbonitrile
(3S,4S)-1-[2-(1-methylpiperidin-4-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1,5-dimethyl-4-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(6-methylpyridin-2-yl)-4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
N-(cyclopropylmethyl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
1-(cyclopropylmethyl)-5-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 4-oxo-4-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)butanoate
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)[(3-methylquinoxalin-2-yl)methyl]amine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-pyrazol-4-yl)butan-1-one
N-methyl-3-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
3-butyl-4-(2,6-difluorobenzenesulfonyl)-1-methylpiperazin-2-one
4-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]propan-1-one
N-(1,2,3-thiadiazol-5-yl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[2-(quinolin-8-yloxy)ethyl]amine
2-[4-(azocan-1-ylmethyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
4-[5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-yl]morpholine
2-[(4-methanesulfonylphenyl)methyl]-2,8-diazaspiro[4.5]decane
2-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
3-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}phenol
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-(1-{1-[(2,4,6-trifluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
(1R,9S)-5-amino-3-(5-fluoro-2-methoxyphenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
N-(cyclopropylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
(1S,4S)-2-(3-chlorophenyl)-5-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[1-(1-{[4-(benzyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
N-(4-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}phenyl)acetamide
4-[(3,5-dimethoxyphenyl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
N-[(4-fluorophenyl)methyl]-3-[1-(pyridazine-4-carbonyl)piperidin-4-yl]propanamide
4-[6-(pyridin-3-yl)pyrimidin-4-yl]morpholine
(3R,4R)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-cyclobutyl-3-methylpiperidin-4-ol
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
ethyl 4-[4-(4-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
5-(3-{[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole