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8-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-imidazole-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-[(3-fluoro-4-methoxyphenyl)methyl]quinolin-8-amine
6-methoxy-N4-methyl-N4-(quinolin-5-ylmethyl)pyrimidine-2,4-diamine
2-(4-fluoro-3-methylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
methyl[(1-{1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]amine
2-benzyl-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
3-chloro-N-cyclopentyl-4-({1-[2-(methylamino)acetyl]piperidin-4-yl}oxy)benzamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidine
2-(3-chloro-4-hydroxyphenyl)-1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]ethan-1-one
4-[(4-methyl-5-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-chloro-4-{[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]methyl}phenol
5-chloro-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
9-[(2R)-2-amino-4-methylpentanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-1-(1,4-dithiepan-6-yl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-methyl-3-phenyl-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N,1,3,6-tetramethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-[2-amino-6-(2-chlorophenyl)-3-cyanopyridin-4-yl]-1H-pyrazole-3-carboxylate
4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-4-oxobutane-1-sulfonamide
4-[4-(4-methoxyphenoxy)piperidin-1-yl]-4-oxobutane-1-sulfonamide
N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
methyl 3-[(3S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]propanoate
N,1-dimethyl-3-(2-methylpropyl)-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-propyl-4-(pyridine-3-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
6-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-1-methyl-1H-indole
2-(2,6-dichlorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-[4-(3-fluorophenyl)phenyl]-N-(1H-imidazol-2-ylmethyl)piperidin-4-amine
3-acetyl-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-(2-aminoethyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
2-(1-methylpyrrolidin-3-yl)-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-(furan-2-ylmethyl)piperidine-1-carboxamide
(2S)-1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidine-2-carboxamide
4-[4-(piperidin-1-ylmethyl)benzoyl]-1,4-oxazepane
2-(3,5-dimethoxyphenyl)pyridine-4-carbonitrile
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(quinolin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(ethyl)(pyridin-3-ylmethyl)amine
6-fluoro-2-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinoline
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclohex-3-ene-1-carboxamide
3-[6-(thiomorpholin-4-yl)pyridazin-3-yl]benzonitrile
1-(but-3-enoyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
3-(2-{[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}ethoxy)benzoic acid
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(piperidin-1-yl)ethyl]acetamide
1-(4-{2-[4-(dimethylamino)azepan-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one