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5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-(propan-2-yl)pyrimidin-2-amine
1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
2-({6-[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-3-(4H-1,2,4-triazol-3-yl)piperidine
(1R,5R)-3-(5-ethylthiophene-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-butyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
4-oxo-4-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]butanamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
2-(6-chloro-2-fluoro-3-methylphenyl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
(3S,4S)-1-[(3-methylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
3-[(7-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}thiomorpholine
1-ethyl-4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(5-ethylpyridin-2-yl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
N-cyclopropyl-1-{1-[2-(4-hydroxyphenyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
{[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
4-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-methylpyrimidine
3-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydroquinoxalin-2-one
6-methyl-5-{5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[1-(2-phenylethyl)piperidin-3-yl]pyridine-4-carboxamide
1-cyclopentyl-4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-1,4-diazepane
1-[(3-fluorophenyl)methyl]-6-methyl-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
7-(1,3-benzothiazol-2-yl)-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(1-methylcyclohexanecarbonyl)-decahydro-1,6-naphthyridin-2-one
3-{3,5-dimethyl-1-[5-(methylcarbamoyl)furan-2-yl]-1H-pyrazol-4-yl}propanoic acid
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
methyl 1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
(2S,4R)-4-(4-fluorobenzamido)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-2-carboxamide
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,5,6-trimethyl-1,2-dihydropyridin-2-one
6-methoxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidin-4-amine
2-({4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)pyridine
2-ethyl-9-[(6-fluoroquinolin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(2,6-difluoro-3-methylphenoxymethyl)-1,2,4-oxadiazol-3-yl]pyrazine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2-fluorophenyl)methyl]benzamide
3-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}propanamide
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-(4-{[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
1-(cyclohexylmethyl)-N-[(2-methyl-1H-indol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
3-{[(2,5-difluorophenyl)methyl]amino}-N-(thiophen-2-ylmethyl)propanamide
8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2,3-dihydro-1H-inden-1-yl)-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
4-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile
[(1R,3S,3aS,6aR)-3-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-5-ethyl-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,2,3-trimethylbenzamide
1-(2-methoxyacetyl)-N-[(4-phenylphenyl)methyl]piperidine-3-carboxamide
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)propanamide