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N-methyl-N-[1-(pyridin-3-yl)pentyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-chlorophenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2R)-2-hydroxy-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
4-chloro-1-ethyl-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}benzamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-methoxyethyl)acetamide
2-chloro-4-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
4-methoxy-N-{2-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
7-(1,3-benzothiazol-2-yl)-4-[(2,5-dimethoxyphenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1-(furan-2-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
N-({4-hydroxy-1-[(2E)-3-phenylprop-2-en-1-yl]azepan-4-yl}methyl)morpholine-4-carboxamide
1-(2-aminopyrimidin-4-yl)-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-chloro-2-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carbonyl)phenol
[(5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]dimethylamine
2-(4-methanesulfonylpiperazine-1-carbonyl)-5-methoxy-1-methyl-1H-indole
N-(4-butylphenyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
2-amino-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-(3-methylbut-2-en-1-yl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methanesulfonamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide
N-(butan-2-yl)-N-[(3-methylthiophen-2-yl)methyl]-1H-imidazole-5-carboxamide
N-methyl-2-(3-phenylpropyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{[5-(1-benzylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
6-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
(1S,3R)-3-amino-N-[2-(benzyloxy)ethyl]cyclopentane-1-carboxamide
5-(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
(2R)-2-(methoxymethyl)-N-[4-(4-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
(4aS,7aR)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-benzyl-3-ethyl-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-1,4-diazepan-5-one
4-(3-{3-[3-(5-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
N-(3-ethoxypropyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
(3S,4R)-3-benzyl-4-methyl-1-(2-methylpyrimidin-4-yl)piperidin-4-ol
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1H-indazole-3-carboxamide
(1R,5S,6R)-3-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
4-[3-(6-hydroxy-1,4-oxazepan-4-yl)-3-oxopropyl]-N-methylbenzene-1-sulfonamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2,2-diphenylacetamide
N-cyclopentyl-6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(1R,5S,6S)-N-tert-butyl-3-{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-(1-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)pyrimidin-2-amine
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
(2S,4S)-4-[2-(dimethylamino)acetamido]-N-ethyl-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
[3-(3-methoxypropyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]methanol
(1s,4s)-4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}cyclohexan-1-amine
(1S,5R)-6-(2-phenylethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane