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1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
3-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(1S,8R)-4-amino-6-(5-cyano-1-methyl-1H-pyrrol-3-yl)-3-azatricyclo[6.2.1.02,7]undeca-2,4,6-triene-5-carbonitrile
4-(pyrimidin-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazine-2-carboxylic acid
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-(oxan-2-ylmethyl)pyrimidin-2-amine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
6-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-[(2-methoxyphenyl)methyl]urea
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-methyl-N-(4-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]carbamoyl}phenyl)furan-3-carboxamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]urea
N-[2-(1,3-benzoxazol-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
3-[1-(6-ethylpyrimidin-4-yl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-N-propyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
3-(2-chlorophenyl)-5-(cyclohex-3-ene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
5-(2-cyclopentylacetyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][2-methyl-2-(piperidin-1-yl)propyl]amine
methyl 4-[4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-4-oxobutanoate
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(1H-imidazol-2-yl)piperidine
2-[(2S)-2-aminopropanoyl]-N-[(4-chlorophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-(1-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazole-5-carbonyl}piperidin-2-yl)ethan-1-ol
3-[5-(2-methyl-4-phenylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]pyridazine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
(1S,5R)-6-(2-cyclopropylpyrimidine-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 3-[(2,5-dimethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-(dimethylamino)ethyl]-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-2-one
2-benzyl-5-(4-methyl-3-phenylpiperazine-1-carbonyl)-1,3-benzoxazole
methyl 4-methyl-3-({[3-(1H-1,2,4-triazol-1-yl)propyl]carbamoyl}amino)benzoate
(2S,4S)-4-{4-[(N,3-dimethylbut-2-enamido)methyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
N-{[(3S,4S)-3-hydroxy-1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}naphthalene-1-carboxamide
4-(1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carbonyl)morpholine-2-carboxylic acid
(2H-1,3-benzodioxol-4-ylmethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
(3S,5S)-1-(2-phenylethyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4,6-dimethylpyrimidine
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]furan-2-carboxamide
1-{4-methyl-2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-5-yl}ethan-1-one
1-{4-[(4,4-dimethylpiperidin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
3-({4-[2-(1-phenylethyl)-1H-imidazol-1-yl]piperidin-1-yl}methyl)pyridine
(3S,4R)-1-(3,5-difluoropyridine-2-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one
2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxylic acid
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(furan-2-yl)-3-phenylpropyl]propanamide
(2S,4R)-4-amino-N,N-diethyl-1-(3-fluoropyridine-2-carbonyl)pyrrolidine-2-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)amine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide