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3-methyl-8-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine
N-[(5-ethylpyridin-2-yl)methyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-{4-[2-(pyridin-2-yl)ethyl]phenyl}-3-[2-(pyrrolidin-1-yl)ethyl]urea
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]thiomorpholine-4-carboxamide
2-[8-(furan-2-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-methyl-4-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
2,3,5,6-tetramethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
[1-benzyl-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl](phenyl)methanol
N-(furan-2-ylmethyl)-4-(1H-pyrazol-3-yl)-N-(pyridin-4-ylmethyl)benzamide
2-({2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
(3S,7S,8aS)-7-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3R)-1-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
[3-(cyclopropylmethyl)-1-[3-methyl-4-(morpholin-4-yl)benzoyl]piperidin-3-yl]methanol
5-cyclobutanecarbonyl-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4S)-3,3,4-trimethyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-ol
1-(2-chloro-5-acetamidobenzoyl)piperidine-2-carboxylic acid
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N,N-dimethylpyrrolidin-3-amine
(3R,4R)-4-(azepan-1-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-ol
5-[2-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
(4aR,7aS)-1-methyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-5-{2-[3-(pyrrolidine-1-carbonyl)phenyl]phenyl}-1,3,4-oxadiazole
[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]methanol
1,3-dimethyl-5-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-1,4-diazepane
[4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)morpholin-2-yl]methanamine
4-(2-phenylphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-(oxan-4-yl)piperidine-3-carboxamide
3-[(3R,4S)-1-(3-chloro-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[3-(propan-2-yl)-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-(6-methoxynaphthalen-2-yl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}morpholine
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
1-(3-methyl-1,2-oxazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}-N,N-dimethylethane-1-sulfonamide
(2R,6S)-4-{1-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,6-dimethylmorpholine
N-benzyl-N-(2-hydroxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-(9-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3,9-diazaspiro[5.5]undecan-3-yl)-2-methylpropan-1-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)propanamide
methyl 8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
2-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-chlorophenyl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
methyl({1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-4-ylmethyl)amine
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
3-({[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine