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(2R)-N1-(2,3-dimethylquinoxalin-6-yl)pyrrolidine-1,2-dicarboxamide
3,3,3-trifluoro-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
3-acetamido-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
N-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
1-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-3-phenylpyrrolidin-3-ol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
6-[(3,4-dimethylpiperazin-1-yl)methyl]pyridine-2-carboxylic acid
methyl 2-[3-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-indol-1-yl]acetate
2-chloro-N-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(3-{[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-phenyl-1,2-oxazole-3-carboxamide
5-acetyl-6-methyl-3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
(2-{2-[1-(1H-1,3-benzodiazole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
5-[2-(4-chlorophenyl)-1H-imidazol-1-yl]-1H-1,2,3-benzotriazole
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
(3S,4R)-3-methoxy-1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-4-amine
1-{2-[1-(1H-imidazol-2-ylmethyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
2-amino-4-{[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]amino}quinazoline-6-carboxylic acid
(3S,7S,8aS)-7-[({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)amino]-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxo-N-phenylacetamide
3-[2-(piperidin-2-yl)ethyl]-5-(pyrimidin-2-yl)phenol
1-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}imidazolidin-2-one
1-ethyl-N-(2-hydroxyethyl)-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(2-hydroxyethyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[methyl(2-phenylethyl)amino]-N-(piperidin-4-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-(quinolin-6-yloxy)piperidine-4-carboxamide
2,2-dimethyl-6-[2-(3-phenylpropyl)morpholine-4-carbonyl]-3,4-dihydro-2H-pyran-4-one
1-methyl-4-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1H-pyrazole
2-{4-[4-(2-propoxyethyl)piperazin-1-yl]quinazolin-2-yl}ethan-1-amine
5-acetyl-3-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
4-(2-hydroxy-3-methylbutanoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N,N-dimethylpropane-1-sulfonamide
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
3-methoxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazin-2-amine
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(pent-2-yn-1-yl)piperidine
6-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-N-ethylpyridine-3-carboxamide
2-(2-hydroxypropyl)-9-(5-methyl-1,3-oxazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-phenyl-5-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-methoxy-3,5-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
methyl({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
2-(3-methoxyphenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
6-(3,4-dimethylpiperazin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-[2-(4-chlorophenyl)ethyl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-amine
2-(2-aminoethyl)-N-[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]quinazolin-4-amine
7-cyclopentanecarbonyl-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]-4-(hydroxymethyl)piperidin-4-ol
1-tert-butyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
2-({[2-(2-fluorophenoxy)pyridin-3-yl]methyl}amino)-6-methylpyridine-3-carbonitrile