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1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-[2-(methylamino)ethyl]piperidine-3-carboxamide
N-cyclopentyl-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-(2-aminopyrimidin-4-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
2-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-4-methylphenol
8-(2-hydroxy-4-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2,6-dimethyl-N-(pyridin-4-ylmethyl)quinoline-3-carboxamide
1-methyl-1'-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-[1-(2-hydroxybutyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chloropyridine-4-carboxamide
3-(1-methanesulfonylpiperidin-4-yl)-N-(3-methylphenyl)propanamide
(1S,5R)-3-cyclobutanecarbonyl-6-(2,6-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
12-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
6-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl]methanol
N-(2-fluorophenyl)-3-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}propanamide
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-2-(thiophen-3-yl)acetamide
N-cyclopropyl-1-{2-[1-(2,4-dimethoxybenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxyphenol
6-[4-(2-chlorophenoxy)piperidin-1-yl]pyrimidin-4-amine
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-(1H-pyrazole-4-carbonyl)piperidine-4-carboxylate
1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
N-{3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-4-methylbenzamide
1-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)azepan-2-one
2-(3-hydroxypropyl)-8-(8-methoxyquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-5-[5-(5-methyl-4,5,6,7-tetrahydro-2H-indazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-[1-(2-phenylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](2-methoxyethyl)amine
N-[(2,4-difluorophenyl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(3aS,6aS)-5-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}-1-methyl-octahydropyrrolo[3,4-b]pyrrole
5-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-acetyl-N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1,4-diazepane-1-carboxamide
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-(3-phenylpropyl)propanamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
[2-(2-ethoxyphenoxy)ethyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-4-carboxamide
1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-[1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide
1-(4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(2-chlorophenyl)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-1,2,3-triazole-4-carboxamide
[(3,5-dichloropyridin-4-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
3,5-dimethoxy-2-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}benzoic acid
2-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}benzoic acid
4-[1-(3-phenylbutyl)azetidin-3-yl]morpholine
({4-[1-(furan-3-ylmethyl)pyrrolidin-2-yl]phenyl}methyl)dimethylamine
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-(naphthalen-1-ylmethyl)-4-{[(trimethylpyrazin-2-yl)methyl]amino}pyrrolidin-2-one
N-cyclobutyl-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide