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1-(azocan-1-yl)-3-(2-methoxy-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
(2R,6R)-11-methoxy-4-(3-methoxypropyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1,9-dimethyl-4-[2-(pyrrolidin-1-yl)benzoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(2-methylphenyl)-4-(oxolan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
2-methyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)propan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methoxybenzamide
3-({4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-1-yl}methyl)benzonitrile
8-[(4-hydroxyphenyl)methyl]-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-dimethyl-3-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}benzamide
3-(morpholine-4-carbonyl)-1-propyl-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
(2S,4R)-4-amino-N-[(3-phenoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
4-{5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}-1H-indole
3-[(3R,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
(4R)-N,3-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazolidine-4-carboxamide
(2-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)urea
N-methyl-N-[1-(pyridin-3-yl)ethyl]-1H-1,2,4-triazole-5-carboxamide
8-(4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)carbamoyl)methyl]-1,2,3-oxadiazol-3-ium-5-olate
(2S,4S)-4-amino-N-[2-(2-ethylphenoxy)ethyl]-N,1-dimethylpyrrolidine-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
2-[2-(1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]pyridine
5-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
[(1-cyclopentylpiperidin-4-yl)methyl][(3-methylphenyl)methyl](pyridin-3-ylmethyl)amine
2-methoxy-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
4-(hydroxymethyl)-1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-ol
N-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-4-fluorobenzamide
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1-ethyl-1H-indole
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenylpropanamide
6-cyclobutyl-2-(2-{[4-(propan-2-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-amine
1-(2-{1-[(4-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}ethyl)-1H-pyrazole
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
2-[3-(2,4-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
2-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-1H-imidazole
{[5-(methoxymethyl)furan-2-yl]methyl}(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholine
2-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
N-(3-chloro-4-fluorophenyl)-3-[(3S)-3-acetamidopyrrolidin-1-yl]propanamide
1-(1-benzothiophen-2-ylmethyl)-3-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]urea