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ethyl 4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine-1-carboxylate
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(4-{1-azabicyclo[3.2.1]octan-5-yloxy}-2-methylphenyl)ethan-1-one
methyl 9-[4-(pyridin-4-yl)piperazin-1-yl]-3-azaspiro[5.5]undecane-3-carboxylate
N-[(3S,4R)-4-propyl-1-(2,4,5-trimethylbenzoyl)pyrrolidin-3-yl]methanesulfonamide
3-(2-methoxyethyl)-8-[1-(methylsulfanyl)propan-2-yl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(3S,4R)-1-(6-cyanopyridin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
6-methoxy-N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
ethyl 2-(2-methyl-5-oxo-1,4-diazepan-1-yl)acetate
2-cyclopropyl-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-methyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
6-(1,4-diazepan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(3-methyl-1-benzofuran-2-yl)methyl]amino}methyl)piperidin-2-one
4-{[5-(2-fluorophenyl)furan-2-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]oxolane-3-carboxamide
N-[4-(1,3-thiazol-2-yl)phenyl]methanesulfonamide
9-(3-methanesulfonylpropanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]pyridine-4-carboxamide
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[(3-methylphenyl)methyl]piperazine
[(5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-2-ethylfuran-3-yl)methyl]diethylamine
6-(2,5-dimethylfuran-3-yl)-2-(4-{[(3-hydroxypropyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-ethyl-N-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
N-(2,4-dimethoxyphenyl)-4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidine-1-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-chloro-N-{2-[(2,2-dimethyloxan-4-yl)formamido]ethyl}benzamide
1-(azocan-1-yl)-3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)propan-1-one
5-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[2-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-2-oxoethyl]-1λ6-thiane-1,1-dione
5-[1-(benzenesulfonyl)cyclopropyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-(pyridin-3-yloxy)acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-phenylmethanesulfonamide
5-cyclopropanecarbonyl-1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-chlorophenyl)methyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
(3S,4S)-1-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]piperidine-3,4-diol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
(3R,4S)-1-(3,5-dimethyl-1H-indole-2-carbonyl)-4-phenylpyrrolidin-3-amine
2-{1-cyclopentyl-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1'-(4-aminopyrimidin-2-yl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-[(3R,4S)-3-(2-carboxyethyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(5-methylhexan-2-yl)-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
(3-{2-[1-(2-ethylpyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
7-chloro-4-methyl-2-[3-(pyridin-4-yl)azetidin-1-yl]quinoline
(2S,4R)-4-amino-N,N-diethyl-1-[5-(4-methylphenyl)furan-2-carbonyl]pyrrolidine-2-carboxamide