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4-(piperidin-3-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
4-methyl-1-{[5-(3-methyl-1H-1,2,4-triazol-5-yl)furan-2-yl]methyl}piperidine
ethyl 4-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}piperidine-1-carboxylate
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
(3S,4S)-1-(2-methyl-1,3-thiazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-methanesulfonamidoacetamide
(1R,2S,4R)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
N,2,3-trimethyl-N-[1-(pyridin-3-yl)pentyl]quinoxaline-6-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidin-3-yl]acetamide
[(4-{[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
4-[2-(5-fluoro-2-methoxyphenyl)pyridine-4-carbonyl]morpholine
methyl (3aS,6aS)-2-[(4-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
1-[(5-chlorofuran-2-yl)methyl]-4-(4-fluorophenoxy)piperidine
5-(benzylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,5S)-5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpyrrolidin-3-amine
1-[3-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)phenyl]ethan-1-one
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-5-methylpyrimidin-4-amine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
(3S,4R)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-[4-(ethanesulfonyl)piperazin-1-yl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
1-(2-methoxyacetyl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}piperidine-3-carboxamide
(1R,3S)-7-(3,5-dimethyl-1H-indole-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylthiophene-2-carboxamide
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
1-{1-[(3,5-difluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
2-amino-3-ethyl-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
9-(dimethyl-1,3-oxazole-5-carbonyl)-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(5-ethylfuran-2-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
2-(2-methoxyethyl)-9-(4-oxo-4-phenylbutyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-fluorophenyl)ethyl]-2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]acetamide
3-(thiomorpholine-4-sulfonyl)-5-(1H-1,2,4-triazol-1-yl)benzoic acid
5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}-3-(propan-2-yl)urea
N-[1-(thiophen-3-yl)propan-2-yl]pyridazine-4-carboxamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-(oxolan-3-yl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
N-(4,6-dimethylpyridin-2-yl)-3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)benzamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
1-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[methyl(2-phenylethyl)amino]-2-(pyridin-2-ylmethyl)-2,3-dihydropyridazin-3-one
1-methyl-4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
(2S,4S)-N-ethyl-4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
N-[2-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)thiophen-3-yl]acetamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
[(3aS,6aS)-2-(2-amino-5-methylpyrimidin-4-yl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol