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ethyl 5-[({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)carbamoyl]-1H-imidazole-4-carboxylate
(1S,5R)-3-benzoyl-N-(2-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N,N-dimethyl-1-{5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-amine
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,4-triazol-3-amine
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(2-methoxyethyl)-2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
4-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-(propan-2-yl)pyridine-2-carboxamide
2-cyclohexyl-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
4-methyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
(1S,5R)-3-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[2-(diethylamino)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)ethane-1-sulfonamide
3-chloro-5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridine
4-(3-ethyl-3-methylpiperidine-1-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
4-(2-aminophenyl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
7-(propan-2-yl)-2-(quinoxalin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
4-(3-methoxypropyl)-11-(4-phenylpiperazin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[1-(4-chlorophenyl)cyclobutyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
6-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methylpropyl)piperidin-4-amine
1-methyl-3-{4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-acetyl-N-(2,2,7-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)piperidine-4-carboxamide
{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
3-methyl-N-(1-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
1,5-dimethyl-4-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[2-(3-chlorophenyl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
4-phenyl-N-(3-{4-[4-(pyridin-3-yloxy)piperidin-1-yl]piperidin-1-yl}phenyl)butanamide
3-[(2-cyclopentyl-1H-imidazol-1-yl)methyl]-1-methanesulfonylpiperidine
1-(2-ethoxyethyl)-N-[(2-methylpyridin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-phenoxy-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}butanamide
3-(2-hydroxyphenyl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{spiro[2.5]octan-1-ylmethyl}propanamide
2-amino-4-(1H-indol-3-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-[2-(ethylsulfanyl)phenyl]-4-(thian-4-yl)piperazine-1-carboxamide
8-chloro-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylquinoline-2-carboxamide
3-hydroxy-N-{2-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]ethyl}pyridine-2-carboxamide
(3aR,5S,6S,7aS)-2-[(5-butylthiophen-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(piperidin-1-yl)pyrimidine
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1H-1,2,3-benzotriazole-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
5-(morpholin-4-ylmethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}furan-3-carboxamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-methyl-1,3-thiazole