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N-[(3R,4R)-3-hydroxy-1-(2-hydroxy-5-methylbenzoyl)piperidin-4-yl]pyridine-2-carboxamide
(3R,5S)-1-benzyl-5-(3-fluorophenoxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
4-({[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
3,3-dimethyl-1-({5-[2-methyl-2-(pyrrolidin-1-ylmethyl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-[2-(3-methylpyridin-2-yl)ethyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
2-[(4-fluorophenyl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-aminoethyl)-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}-1H-1,2,3-triazole-4-carboxamide
1-{3-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-chloro-4-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]butan-2-ol
N-[(5-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
2-(dimethylamino)-N-[3-(pyridin-3-yloxy)propyl]-2,3-dihydro-1H-indene-2-carboxamide
6-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)-1,2,3,4-tetrahydroquinolin-2-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-azaspiro[5.5]undecan-9-amine
2-(2-chlorophenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-2-methyl-2H-1,2,3,4-tetrazole
(2S,3R)-3-hydroxy-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}butanamide
[(3R,4R)-1-(5-methylthiophene-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
methyl 2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-2-methylpropanoate
N-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
[1-(1H-pyrazol-3-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
[(2-fluorophenyl)methyl](methyl){[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(4aS,8aS)-2-(4-ethoxy-3-methylbenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{3-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]propyl}piperidine-3-carboxamide
[(2S,6S)-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(2S,4S)-4-(2-cyanobenzamido)-N-ethyl-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
(3R,5S)-1-benzyl-N-butyl-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
5-ethyl-2,3-dimethyl-N-[(3-methyloxetan-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-cyclopropyl-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
4-methyl-9-(4-phenylbenzoyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-N-(1-benzothiophen-5-ylmethyl)-3-(1H-imidazol-4-yl)propanamide
N,1-dimethyl-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,6-dihydropyridine-3-carboxamide
3-(2-methyl-1-benzofuran-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-[methyl(phenyl)amino]-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1,7-dimethyl-1H-indole-2-carboxamide
2-methoxy-5-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
N3-cyclooctyl-N5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]-6-methylpyridine-3-carbonitrile
methyl[1-(pyrimidin-4-yl)ethyl]{[2-(trifluoromethyl)phenyl]methyl}amine
1,5-dimethyl-4-[3-methyl-1-(2-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
7-amino-4-[3-(ethoxymethyl)-4-methoxyphenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-(1-{6-[(2-methoxyethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
1-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-4-yl]pyrrolidin-2-one
4-benzyl-3-ethyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,4-diazepan-5-one
N-[1-({[2-(furan-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
3-({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione