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1'-(1H-indol-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{4-[4-(2-methylphenoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
4-[(3-fluorophenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
2-(benzyloxy)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
4-[(E)-2-phenylethenyl]benzamide
N3-(1,3-benzothiazol-2-ylmethyl)-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
N-[(1R,2R)-2-(benzyloxy)cyclohexyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1H-1,2,3-benzotriazol-5-yl)-5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-N-(2-methoxy-5-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-(4-methoxyphenyl)-N,N,2-trimethyl-3-oxopiperazine-1-sulfonamide
4-(1-aminocyclopropanecarbonyl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(6-methoxypyridin-3-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
3-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-[({1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N,N-diethyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazine-1-sulfonamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-ethylpyrimidine
4-({3-[methyl(phenyl)amino]propyl}sulfamoyl)-N-(propan-2-yl)benzamide
(4aS,8aR)-6-(2-amino-6-methylpyrimidin-4-yl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-2-oxo-N-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(hydroxymethyl)piperidine-1-carbonyl]piperidin-2-one
1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-methyl-6-(2-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}ethyl)pyrimidin-4-ol
2-{4-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-amido]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
4-[3-(3-methoxypiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
2-(1H-indol-3-yl)-1-[2-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
5-(1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2-methyl-5-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrazine
(2R)-2-cyclohexyl-2-hydroxy-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
(1R,5S,6S)-3-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-6-(4-methyl-1,4-diazepane-1-carbonyl)-3-azabicyclo[3.1.0]hexane
3-(3-{[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]methyl}-1H-indol-1-yl)propanamide
4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]morpholine
2-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3S,4R)-1-[3-(hydroxymethyl)quinolin-2-yl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-{6-hydroxy-4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
7-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-2-cyclopropyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
N,N-dimethyl-5-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)pyrimidin-2-amine
5-[4-(aminomethyl)piperidin-1-yl]-2-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,3-dihydropyridazin-3-one
1-[(4-methanesulfonylphenyl)methyl]-4-(3-methylpyridin-2-yl)piperazine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(morpholin-4-yl)propanamide
1-cyclohexyl-4-[(3S,4S)-4-hydroxy-1-(4-methoxybenzoyl)pyrrolidin-3-yl]piperazin-2-one
8-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyridin-2-amine