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1-methyl-8-(4-methylpyridine-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-1-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-[2-(4-hydroxypiperidin-1-yl)ethyl]-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-acetyl-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-4-carboxamide
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[(2-methoxyphenyl)methyl]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
1-(1H-pyrrole-2-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-methanesulfonyl-4-[4-(pyridin-3-yl)pyrimidin-2-yl]-1,4-diazepane
2-(2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
(1-{[methyl(trimethylpyrimidin-4-yl)amino]methyl}cyclobutyl)methanol
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
3-{[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
methyl (2S,4S)-4-[3-(4-methylphenyl)propanamido]-1-(propan-2-yl)pyrrolidine-2-carboxylate
3-(4-benzyl-1H-pyrazol-5-yl)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
1-[(5-acetylthiophen-3-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-[3-(3-ethoxy-5-fluorophenyl)phenyl]-5-methyl-1,3,4-oxadiazole
2-{4-methyl-6-[(oxan-2-ylmethyl)amino]pyrimidin-2-yl}phenol
3-[(3,4-dimethoxyphenyl)methyl]-5-(1H-pyrrol-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-(1H-imidazol-1-yl)-1-{4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
(3S,7S,8aS)-7-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl N-{2-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-2-oxoethyl}carbamate
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
4-(2,5-dihydro-1H-pyrrol-1-yl)-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-benzothiazole-6-carboxamide
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
2-methyl-8-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
6-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carbonitrile
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-hydroxy-4-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]benzamide
N-{2-[5-(5-methyl-1H-indol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetic acid
N-[2-(3-methylphenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(4-fluorophenyl)-2-hydroxy-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-2-amine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[(2,3-difluorophenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
N-[1-(4-fluorophenyl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
4-(3,5-difluoro-4-methoxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
2-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(pyridin-4-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
1-ethyl-N,3-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}benzamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-2-(2-oxopyrrolidin-1-yl)acetamide
(3R,4R)-4-(azepan-1-yl)-1-[(3-chloro-4-ethoxyphenyl)methyl]piperidin-3-ol
7-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylpentanamide