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1-[3-({3-[(4-methoxyphenyl)amino]piperidin-1-yl}methyl)phenyl]ethan-1-one
N-[1-(methoxymethyl)cyclopentyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-methyl-5-[4-(pyrrolidin-2-yl)phenyl]furan-2-carboxamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
2-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-N-(isoquinolin-5-ylmethyl)-N,4-dimethylpyrimidine-5-carboxamide
1-(cyclopropylmethyl)-5-(2-acetamidoacetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4aS,8aR)-1-(3-aminopropyl)-6-(3-chlorothiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(1R,3S)-7-[3-(methylsulfanyl)propyl]-7-azaspiro[3.5]nonane-1,3-diol
5-methoxy-N-[2-(thiophen-2-yl)ethyl]-1-oxa-9-azaspiro[5.5]undecane-9-carboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(3-ethoxyphenyl)methyl](2-methoxyethyl)amine
methyl 2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1-methyl-1H-1,3-benzodiazole-5-carboxylate
1-[2-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-methyl-1H-indole
N-butyl-1-[2-(3,4-dimethoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
methyl 6-[(4-methoxy-3-methylphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(cyclohex-1-en-1-yl)ethyl]-1,3-dimethyl-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
(1S,5R)-3-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(5-fluoro-2-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(2R,3R,6R)-3-(4-methylphenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-chloro-2-{[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}-1H-1,3-benzodiazole
(2S)-2-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidine-1-carboxamide
2-{5-[2-(benzenesulfonyl)ethyl]-1-cyclohexyl-1H-1,2,4-triazol-3-yl}acetamide
N-[(2S,4R,6S)-2-benzyl-6-(quinolin-3-yl)oxan-4-yl]acetamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
1,5-dimethyl-2-phenyl-4-[(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2,3-dihydro-1H-pyrazol-3-one
1-(4-{1-[(4-methoxyphenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)butan-2-ol
4-[1-(2,3-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
10-methoxy-5-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
4-benzyl-3-ethyl-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
N-(2-ethylphenyl)-3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(3,4-dichlorophenyl)-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]morpholine
N-(2-methoxyethyl)-1-[1-(3-methylbenzoyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-{2-hydroxy-3-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
4-{[5-(1-benzoylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
1-[3-(propan-2-yloxy)propyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
11-[(2,3-dihydro-1H-inden-2-yl)amino]-4-[2-(2-fluorophenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
5-methyl-3-(4-phenyl-1H-imidazol-5-yl)-1H-indole-2-carboxylic acid
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
5-{[2-(3-chlorophenoxy)ethyl](methyl)carbamoyl}-1H-imidazole-4-carboxylic acid
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
4-{2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N'-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)ethanediamide
N3-cyclooctyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(5-{[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
N-[(2,4-difluorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine