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N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-{1-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-oxoimidazolidine-4-carboxamide
N-(1-methyl-1H-1,2,4-triazol-3-yl)-3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)benzamide
6-chloro-5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}imidazo[2,1-b][1,3]thiazole
2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
1-(2,3-dimethylphenyl)-4-{[4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
2-(4-chloro-2-methylphenoxy)-N-(oxolan-3-yl)acetamide
1-[4-(azetidin-1-ylmethyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
methyl 3-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoate
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
methyl 3-[(3-ethoxyphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-[(4-fluorophenyl)methyl]-2-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}piperidin-2-one
(1R,3S)-3-(2-hydroxyethoxy)-7-(5-methoxypyrimidin-2-yl)-7-azaspiro[3.5]nonan-1-ol
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-ethyl-2-(1-ethylpiperidin-4-yl)-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]acetamide
N-methyl-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(2-methyl-1H-imidazol-1-yl)propanamide
2-ethyl-4-phenyl-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}quinazoline
[(4aS,8aR)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(2-fluorophenyl)methyl]-3-{1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}propanamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-(4-methylpiperazin-1-yl)pyrimidine
2-(2-methoxy-5-methylphenyl)-2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
3-{[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-3-(3-methoxypropyl)piperidine
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholin-2-yl]ethan-1-ol
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
N-(2-{7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
2-[4-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
{1-[4-(4-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
2-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-cyclohexyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N-ethylbenzamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
8-[4-(1H-pyrazol-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
9-(cyclopropylmethyl)-4-(4-ethenylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(5-methyl-1,2-oxazol-3-yl)-2-[2-(propan-2-yloxy)propanoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1,2-benzoxazole
4-(2-aminopyridine-4-carbonyl)-7-(1-benzothiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1,2,3,4-tetrahydroquinolin-2-one
2-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}pyridine