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1-(3-{1-[(2-methoxyphenyl)methyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({1-[(3,5-difluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-2,2-difluoroacetamide
5-amino-N-[(5-fluoro-2-methylphenyl)methyl]-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
N-(2-acetamidoethyl)-3-(2-methylphenyl)-3-phenylpropanamide
ethyl 3-[(4-fluorophenyl)methyl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylate
5,7-dimethyl-2-(2-methylpyrimidin-5-yl)-4-(morpholine-4-carbonyl)quinoline
(1R,5S,6S)-6-(3,3-diphenylpiperidine-1-carbonyl)-3-azabicyclo[3.1.0]hexane
3-{1-butyl-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazol-3-yl}-1H-indole
[(3R,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(oxane-4-carbonyl)piperidin-3-yl]methanol
3-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-benzyl-N-methylpropanamide
2-[({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-2-methylpropanamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
2-{5-[(oxan-2-ylmethoxy)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}pyridine
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-2-(2-oxopiperidin-1-yl)acetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(methylsulfanyl)pyridine-3-carboxamide
5-methyl-5-phenyl-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-2-one
1-(4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
1-[(3,5-difluorophenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
(3aR,5R,6S,7aS)-2-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-octahydro-1H-isoindole-5,6-diol
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(2,4,4-trimethylpentan-2-yl)piperidine-1-carboxamide
1-(9H-fluoren-2-ylmethyl)-3-(pyrrolidin-1-yl)pyrrolidine
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-{5-[(4-methoxy-3-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
2-chloro-N-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
3-(pentan-2-yl)-8-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopropyl-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]acetamide
N5-cyclopropyl-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(4-methoxybenzoyl)piperidine
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(phenylsulfanyl)ethyl]piperazine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
(1R,5R)-6-(cyclopropylmethyl)-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-benzyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-[2-(methylsulfamoyl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N-{3-[5-(aminomethyl)-2-fluorophenyl]phenyl}acetamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(4-butanamido-3-methoxyphenyl)-5-chloro-2-oxo-1,2-dihydropyridine-3-carboxamide
1-methyl-3-(propan-2-yl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-6-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)-1H-indole
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-fluorophenyl)methyl]amine
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]isoquinoline
2-{[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-2H-1,2,3-benzotriazole
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[2-phenyl-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one