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N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-(2-chloro-4-{[methyl({[1-(propan-2-yl)pyrrolidin-3-yl]methyl})amino]methyl}phenoxy)acetamide
N-(3-hydroxy-3-methylbutyl)-N-methyl-1-benzothiophene-2-carboxamide
2-{2-[5-(1-methyl-1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}ethan-1-ol
1-methyl-6-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(2,5-dimethylphenoxy)propyl]-N-methylpyrimidin-4-amine
N-(2-methoxyethyl)-4-(quinolin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aR,8aR)-4-[(2-cyclohexylpyrimidin-5-yl)methyl]-octahydro-2H-1,4-benzoxazine
N-{2-methoxy-4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
(2S,4S)-4-(3,4-dimethylbenzamido)-N-ethyl-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
methyl 1-({3-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]phenyl}methyl)piperidine-2-carboxylate
N,4,6-trimethyl-N-(1,2-oxazol-3-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(2-ethylphenyl)pyridine-2-carbonitrile
4-(2,5-dimethylthiophen-3-yl)-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
3-[({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)methyl]pyridin-2-ol
2-(2-methoxyethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-(cyclohex-3-en-1-ylmethyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(2-{methyl[(3-methylphenyl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
6-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-4-[4-(morpholin-4-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}isoquinoline
2-ethoxy-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[1-(3-methoxyphenyl)propan-2-yl]amine
3-ethyl-1-[2-(thiophen-2-yl)acetyl]piperidine-3-carboxylic acid
1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-3-yl)morpholine
5-methyl-6-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-methyl-3-(5-methylfuran-2-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
6-ethyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-benzyl-8-[(3-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[(2,4,6-trimethylphenyl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
(2S)-2-acetamido-N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(methylsulfanyl)butanamide
ethyl 2-(4-{[3-(2-methoxyphenoxy)azetidine-1-carbonyl]amino}phenyl)acetate
(2S,4S)-N-[(2,5-dimethoxyphenyl)methyl]-4-(furan-2-amido)-1-methylpyrrolidine-2-carboxamide
1-(2-ethylphenyl)-3-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]urea
2-(adamantan-1-yl)-N-[2-(methylsulfamoyl)ethyl]acetamide
1-ethyl-2-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
2-{[3-(dimethylamino)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-(diethylamino)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
5-benzyl-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N,N-dimethyl-5-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-{2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]ethyl}acetamide
(2R,6R)-4-[4-(morpholin-4-yl)butanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-phenylethan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]oxane-4-carboxamide
5-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1,2,4-oxadiazole