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methyl 5-[(3-hydroxypiperidin-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-methoxypyridine-3-carbonitrile
ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
2-[methyl(pyridin-3-ylmethyl)amino]-2-[2-(methylsulfanyl)phenyl]acetic acid
N-{[1-(1-methylpiperidin-4-yl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
1-[2-chloro-4-(1H-pyrazol-1-yl)benzoyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
ethyl 2-[4-(3-methoxybenzoyl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-7-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(1H-pyrrol-1-yl)phenyl]acetamide
6-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
4-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-oxopropyl)-N-methylbenzene-1-sulfonamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-methoxy-5-[({2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}carbamoyl)amino]-N-methylbenzamide
2-{3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-indazole-3-carboxamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-(cyclopropylmethyl)-2,3-dihydropyridazin-3-one
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
3-butyl-1-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-chloropyridin-2-yl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-4-ylmethyl)piperazine
6-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]pyridin-2-amine
2-({4-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N,2,5,6-tetramethyl-N-[(3-methylpyridin-4-yl)methyl]pyrimidin-4-amine
2-hydroxy-5-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)benzoic acid
N-[2-(2,5-dimethylphenoxy)ethyl]-4-acetamido-N-methylbutanamide
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-3-(2-chlorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-[4-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidine
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-(dimethylamino)-N-(3-methyl-1-{7-[3-(methylsulfanyl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
3-{[2-methyl-4-(methylcarbamoyl)butan-2-yl]carbamoyl}benzoic acid
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-benzyl-5-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}pyrimidin-2-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-3-yl)propanamide
N-(4-methoxy-2-methylphenyl)-3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}propanamide
[(2-methoxyphenyl)methyl](prop-2-en-1-yl){[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
4-(1H-imidazol-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-N,N-dimethylethane-1-sulfonamide
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,8aR)-6-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[2-(dimethylamino)ethyl]-5-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
(3aR,5S,6S,7aS)-2-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(3-fluorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
3-[1-(2,5-dimethylbenzenesulfonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
4-ethyl-3-[(1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one