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2-(pyridin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidine-5-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)furan-2-carboxamide
(3S,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine
N-[(2,3-dimethoxyphenyl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(2-fluoro-5-methoxyphenyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetic acid
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
5-phenyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
8-methoxy-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-[methyl(pyridin-2-ylmethyl)amino]-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-(2-ethylpyridin-4-yl)-1H-1,2,4-triazol-3-yl}acetamide
N-{3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,6-dimethyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-(quinolin-5-ylmethyl)furan-2-carboxamide
2-[(2-fluorophenyl)methyl]-6-(pyrrolidine-1-carbonyl)-1,3-benzoxazole
N-[2-(3,5-dimethoxyphenyl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
3-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-[(1S,5R)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(5-phenyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[3-(morpholin-4-yl)propyl]acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
1-{3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-(4-methylphenyl)pyrrolidin-2-one
4-{[5-(1,4-dioxan-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-{4-[8-methyl-2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)quinazolin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
5-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]-1H-1,2,3-benzotriazole
5-(ethylamino)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2,4-triazin-3-amine
N-[(2-ethoxyphenyl)methyl]-N-(furan-3-ylmethyl)cyclopropanamine
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidine
6-(4-chlorophenyl)-N-(2-hydroxyethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
(5S,9aS,9bS)-2-phenyl-5-(3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(oxan-4-yl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-(4-phenyl-1H-imidazol-1-yl)acetamide
2-{[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
2-[2-methoxy-4-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}propan-1-one
2-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carbonyl)pyridine
(3R,4R)-4-cyclobutyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-methylpiperidin-4-ol
N-benzyl-2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-hydroxyethyl)acetamide
5-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-methoxy-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1H-indole-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)acetic acid