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1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
1-(2-methoxy-4-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,4-dithiepan-6-amine
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
4-(4-methylpiperazin-1-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]({[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl})amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 4-(5-{[(3S,4S)-3,4-dihydroxypiperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(5S)-5-{[(1-methanesulfonylpiperidin-4-yl)(pyridin-4-ylmethyl)amino]methyl}pyrrolidin-2-one
3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
N,N-dimethyl-4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-carboxamide
3-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methylphenyl)urea
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(naphthalen-2-yloxy)-1-(trimethylpyrimidin-4-yl)piperidine-4-carboxylic acid
1-(3-methoxybenzoyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-1H-indole
4-[2-(2-chloro-4-methylphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(cyclopropylmethyl)-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(5-methylfuran-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(oxan-4-ylmethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N3-cyclohexyl-N5-(2-hydroxybutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl](pentan-3-yl)amine
8-(2-fluorobenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-ol
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
3-[4-(2-chlorophenyl)piperazine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
4-{1-[2-(furan-2-yl)ethyl]-1H-imidazol-2-yl}quinoline
5-methyl-1'-[2-(1H-pyrazol-1-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
methyl 4-oxo-4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)butanoate
3-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-[3-(4-methanesulfonyl-1,4-diazepan-1-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
(1S,5R)-3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
3-{2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
6-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridine-2-carboxylic acid
3-{1-[(3-chloro-1-benzothiophen-2-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
6-methyl-1-{3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
4-[(pyridin-2-ylmethyl)sulfamoyl]-N-[(3S)-pyrrolidin-3-yl]benzamide
1-(2,4-dimethyl-6-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-1H-pyrazole