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3-{[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
{[4-(2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]methyl}dipropylamine
1-[3-(2-ethylphenoxy)azetidin-1-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
3-(morpholin-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(thiophen-2-yl)ethan-1-one
methyl 3-({5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
4,4,4-trifluoro-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
[(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
3-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]pyridin-2-amine
2-cyclopropyl-8-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-(4-carbamoylpyridin-2-yl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
methyl (2S)-1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidine-2-carboxylate
N-[2-(furan-2-yl)ethyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
2-[(adamantan-1-ylmethyl)({[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
N-[(5-methylpyrazin-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
methyl (1R,3S,3aR,6aS)-1-ethyl-3-(1-methyl-1H-pyrazol-4-yl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-(1-methyl-1H-imidazol-2-yl)-1-[2-(3-methylthiophen-2-yl)ethyl]-4-phenyl-1H-imidazole
4-hydroxy-2-(pyridin-2-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
(2E)-3-(4-methoxyphenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
N-(2-methyl-4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)pyridine-3-carboxamide
11-[4-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-butyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,N-dimethyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
3-{1-azabicyclo[2.2.2]octan-3-yl}-1-[4-(1H-pyrazol-1-yl)phenyl]urea
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-[7-(1H-imidazol-1-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]-3-(oxolan-2-ylmethyl)urea
methyl({[5-(1-methyl-1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})(1,2-oxazol-5-ylmethyl)amine
N-ethyl-1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidine-3-carboxamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[2-(furan-2-yl)-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-hydroxyethan-1-one
4-[(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
3-(5-methylthiophen-2-yl)-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-indole
(2S)-N-(2,3-dihydro-1H-inden-5-yl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
6-methyl-2-(3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
N,N-dimethyl-4-(4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazine-1-carboxamide
N-(pyridin-4-ylmethyl)-2-(trifluoromethyl)pyrimidin-4-amine
5-{4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)methyl]-1,2,3-oxadiazol-3-ium-5-olate
1-(naphthalen-1-ylmethyl)-4-[(thian-4-yl)amino]pyrrolidin-2-one
3-methyl-6-{5-[3-(thiophen-2-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
ethyl 5-[(3-methylquinoxalin-2-yl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,6R)-3-[(5-methylthiophen-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
4-[3-(2-amino-1,3-thiazol-4-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{2-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
4-(1,3-benzothiazol-2-yl)-2-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}phenol
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
(3S,4S)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-cyclopropylpyrrolidine-3-carboxylic acid