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diethyl[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]amine
2-(3-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
2-(5-fluoro-2-methoxyphenyl)-2-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetic acid
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[2-(methylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
2-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]oxane-2-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholine
4-[1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazol-5-yl]quinoline
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]propanamide
3-(2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methylphenyl)-1,3-oxazolidin-2-one
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
3-{1-[(4-methanesulfonylphenyl)methyl]piperidin-2-yl}propanoic acid
5-methoxy-N-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
5-ethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
methyl 4-(5-methyl-4-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}-1,3-oxazol-2-yl)benzoate
ethyl 6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-3-carboxylate
2-ethyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
4-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-(2-{[ethyl(propan-2-yl)amino]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
2-{1-cyclohexyl-4-[(2,6-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{4-[3-(4-methoxyphenyl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
N-(2-methoxyethyl)-1,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
7-[(2,3-difluorophenyl)methyl]-2-propanoyl-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-2-(1,4-oxazepan-4-yl)propanamide
N-cyclopropyl-3-(1H-pyrazol-1-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
4-[4-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-cyclopentyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-5-oxopyrrolidine-3-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
N-butyl-6-cyano-N-(furan-2-ylmethyl)pyridine-3-carboxamide
7-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 5-[({1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}formamido)methyl]furan-2-carboxylate
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-{[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-hydroxy-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-{3H-benzo[e]indole-2-carbonyl}-3,9-diazaspiro[5.5]undecane
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
3,5-dimethyl-4-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(3-methylbutyl)amino]methyl}phenoxy)propan-2-ol
2-amino-4-(2-methoxypyrimidin-5-yl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
N,N-dimethyl-5-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
2-(3-fluorophenoxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
methyl N-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-oxopropan-2-yl)carbamate
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(2-fluorophenyl)propan-1-one
N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-1,3-thiazole-5-carboxamide
N-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
2-methyl-6-(piperidin-4-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-4-amine
N-ethyl-3-(2-methyl-1H-indol-1-yl)-N-(pyridin-4-ylmethyl)propanamide
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(morpholin-3-yl)acetamide