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6-methoxy-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidin-4-amine
5-acetyl-N-[1-(1H-indol-5-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({1-[(3-acetylphenyl)methyl]piperidin-3-yl}methyl)-1-(4-chlorophenyl)cyclopropane-1-carboxamide
5-methyl-1-(2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-cyclopropyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2,6-diamino-4-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
4-methyl-2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
3-{[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[3-(trifluoromethoxy)phenyl]urea
methyl 1-({1-[(2-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperidine-4-carboxylate
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(ethanesulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-({4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethyl]pyrrolidin-2-one
(1R,6S)-9-methyl-3-(5-phenyl-1,2-oxazole-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-[(2R,4R,6S)-2-tert-butyl-6-[3-(1H-pyrazol-1-yl)phenyl]oxan-4-yl]acetamide
9-(1H-indole-5-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
3-fluoro-5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
methyl 4-[(3-{2-[(5-chloro-2-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
6-methyl-3-{[4-(2-phenylethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
4-chloro-2-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-(3,4-difluorophenyl)-1-(2-methylfuran-3-carbonyl)piperidin-3-amine
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-4-phenylbutane-1,4-dione
2-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}propanamide
5-methyl-5-phenyl-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}piperidin-2-one
2-{1-[(2-chlorophenyl)methyl]pyrrolidin-3-yl}benzoic acid
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3,3-trifluoropropanamide
3-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-(2-methylpropyl)-5-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)pyrrolidine-3-carboxamide
3-chloro-N-(2-methoxyethyl)-6-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-amino-3-ethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{4-methoxy-3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}acetamide
2-(2-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(3S,4R)-1-(oxan-4-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}benzonitrile
ethyl 4-{3-[(2-phenylethyl)carbamoyl]phenoxy}piperidine-1-carboxylate
1-{1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-indol-2-one
3-[5-(1,3-benzoxazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(thian-4-yl)piperazine