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3-[(3R,4S)-4-(morpholin-4-yl)-1-(pyrimidin-2-yl)piperidin-3-yl]propan-1-ol
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophen-3-yl)acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
N-(1,4-dioxan-2-ylmethyl)-N,6-dimethyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-(furan-3-ylmethyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
1-(2-phenylphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-one
1-(oxan-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(thiophen-3-yl)acetamide
(2R)-2-amino-3-phenyl-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
1-[1-(1H-indole-6-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
{1-[(2,7-dimethyl-1H-indol-3-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
2-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyridine-4-carboxamide
2-(1-methyl-1H-pyrazol-3-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
N,2,3-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]quinoxaline-6-carboxamide
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-6-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
N-[2-(dimethylamino)-1-phenylethyl]-5-ethyl-2-methylpyrimidin-4-amine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
4-[(2-methyl-1H-imidazol-1-yl)methyl]-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{4-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]morpholin-3-yl}acetamide
(4aS,7aR)-1-(furan-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
(2S,4S)-4-amino-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
1-(2-methoxyethyl)-4-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-({2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(3S,5R)-1-[(3-hydroxyphenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-[3-(4-fluorophenyl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-3-carboxamide
1-cyclohexyl-4-(1H-indol-4-ylmethyl)piperazin-2-one
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
3-cyclopropaneamido-N-[(2-methoxyphenyl)methyl]-4-methylbenzamide
4-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]-N-phenylpiperidine-1-carboxamide
N-ethyl-2,5-dimethyl-N-(oxan-4-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(1-methyl-1H-pyrazol-4-yl)-2-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]pyrimidine
5-(4-chlorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2,4-triazin-3-amine
3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-cyclopentyl-N5-[(2,6-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopentyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(thiophen-3-ylmethyl)acetamide
2-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,3-benzodiazole
{2-[(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-1-yl)methyl]phenyl}methanol
1-(dimethyl-1,3-oxazole-5-carbonyl)-3,3-diphenylpiperidine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxoazonan-1-yl)acetamide