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methyl[(3-methylpyridin-4-yl)methyl][(1-phenyl-1H-pyrazol-5-yl)methyl]amine
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[(3-methylphenyl)methyl]-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decane
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclohexyl-5-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
7-(cyclopropylmethyl)-2-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(4-methoxypyridin-2-yl)methyl]-2-(pyridin-3-yl)acetamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-9H-purin-6-amine
2-(3,4-dimethylphenyl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]oxane-4-carboxamide
5-(1-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[2-(2,6-difluorophenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
2-{5-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[(2,3-dimethoxyphenyl)methyl]-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2E)-N-tert-butyl-3-(1-methyl-1H-pyrazol-4-yl)-N-(thiophen-3-ylmethyl)prop-2-enamide
(4aS,7aR)-1-[(6-chloroquinolin-2-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,6R)-9-[4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{2-[1-(2-chloro-6-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
(3S,9R)-11-[(5-chlorothiophen-2-yl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-(4-methylphenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]-1-(4-methoxyphenyl)-1H-1,2,4-triazole
(2R,6S)-4-[6-chloro-3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-2,6-dimethylmorpholine
4-(hydroxymethyl)-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-4-ol
(2S,4R)-1-benzyl-4-{[(3,4-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
3-({1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
1-[7-(furan-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-3-methoxypiperidine
N-methyl-6-(piperidin-1-yl)-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
6,7-dimethyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole
4-[2-(3,3-diphenylpiperidin-1-yl)ethyl]morpholine
2-(4-chlorophenyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]morpholine
1-(3,5-difluoro-4-methoxybenzoyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(4-methyl-5-{[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
2,7,8-trimethyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]quinoline
2-[3-(2,6-dimethylphenyl)-1H-indazol-1-yl]-N-(1-ethyl-1H-pyrazol-5-yl)acetamide
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
4-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}benzoic acid
5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-2-oxo-N-(prop-2-en-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
8-[2-(1H-indol-3-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
(3aR,6aR)-2-(2-methoxyethyl)-5-(3-methylpyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methoxy-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-phenylpiperidine
3-methyl-7-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(4aS,8aR)-6-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-3-carboxamide