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(1R,3S)-7-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(diphenylmethyl)-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(3-chloro-4-propanamidophenyl)-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
3-chloro-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]pyridine-4-carboxamide
1-(3-chloro-4-propoxybenzoyl)-3-(1H-imidazol-2-yl)piperidine
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-[2-(4-methylphenyl)ethyl]urea
1-[(4-fluorophenyl)methyl]-4-[(2-methyl-6-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
3-[5-(6-ethoxypyridin-3-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyridine-3-carboxamide
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
2-amino-N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[2-(butan-2-yl)phenoxy]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
(2S)-2-amino-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylethan-1-one
3-methyl-8-(1-methyl-1H-indole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-methyl-8-(2-methyl-6-propylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-[({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-(2-methoxyacetyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
[(3R,4R)-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-benzyl-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-carboxamide
N-[3-(2-fluorophenyl)propyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{[5-(1-methoxyethyl)-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2S,4S)-4-amino-N-ethyl-1-[3-(1,2-oxazinan-2-yl)propanoyl]pyrrolidine-2-carboxamide
N-(1-{1-[(2S)-2-acetamido-4-methylpentanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(4aS,7aR)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(5-{[benzyl(4-hydroxybutyl)carbamoyl]amino}-2-fluorophenyl)acetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({[3-(methylsulfanyl)phenyl]methyl})amine
5-(methoxymethyl)-3-[(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
(3R,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1-azabicyclo[2.2.2]octan-3-amine
1-cyclohexyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
N-phenyl-4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}phenol
N-[(4-hydroxy-3-methoxyphenyl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1H-1,3-benzodiazol-2-yl)methanol
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
3-(oxolan-3-yl)-5-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-4-yl}-1,2,4-oxadiazole
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-(2-methylphenyl)urea
(2S)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-acetamido-4-(methylsulfanyl)butanamide
1-{3-[2-(4-fluorophenyl)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
N-[(2S)-2-aminopropyl]-2-cyclopropyl-4-methylpyrimidine-5-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
2-{4-[(3-methylthiophen-2-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
8-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one