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1-methyl-2-(morpholin-4-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
9-(2,6-dimethylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-1-benzyl-N-butyl-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
3-methyl-4-oxo-N-[3-(phenylsulfanyl)propyl]-3,4-dihydroquinazoline-7-carboxamide
methyl 4-{[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]formamido}butanoate
3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3,5,6-tetramethylbenzamide
N4,N4,5-trimethyl-N2-[1-(1-methyl-1H-imidazol-2-yl)butyl]pyrimidine-2,4-diamine
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{2-[1-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-[(8-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
4-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-4H-1,2,4-triazole
2-(2,5-dimethoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
1-cyclohexyl-N3-[(1R)-1-(4-methoxyphenyl)ethyl]-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2-(2-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-{[1-(2-methylpropyl)piperidin-2-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3,4-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-methyl-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(5-fluoro-2-methyl-1H-indol-3-yl)acetamide
1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
6-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-benzyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3-benzoxazole-5-carboxamide
N,2-dimethyl-N-(1H-pyrazol-5-ylmethyl)-3-[(pyridin-3-ylmethyl)amino]benzamide
1-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-[1-(1-benzothiophen-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
6-cyclopropyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyrimidin-4-amine
2-({[2-(furan-2-yl)phenyl]methyl}(methyl)amino)-N,N-dimethylpropanamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidin-4-ol
4-(5-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazole
4-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}-N-phenylbenzamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-[2-(1H-imidazol-1-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-[(2,4-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(phenylsulfanyl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
3-methyl-8-[2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-butyl-3-[(3,4-dimethoxyphenyl)methyl]-5-(oxan-4-yl)-1H-1,2,4-triazole
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
2-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)amino}methyl)benzonitrile
2-{1-[(3-methoxyphenyl)methyl]-4-propylpiperazin-2-yl}ethan-1-ol
N-[4-methyl-3-(4-methylbenzamido)phenyl]-4-sulfamoylbenzamide
N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane