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4-[3-(benzylcarbamoyl)phenoxy]-N-propylpiperidine-1-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(2-methoxyethyl)piperidine
3-chloro-2-(5-chloro-2-methoxyphenyl)pyridine
3-(4-ethyl-1H-pyrazol-5-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(2,6-dimethylpyridin-4-yl)-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{2-[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-({7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
1-(4-benzylpiperidin-1-yl)-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propan-1-one
2-[(3-{[(5-methylpyrazin-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
N-methyl-N-(pyrazin-2-ylmethyl)-1-benzothiophene-2-carboxamide
4-{[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]methyl}-2,6-dimethoxyphenol
(2S,4R)-1-(furan-2-ylmethyl)-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-fluoro-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(3S,4S)-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-hydroxy-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-({1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-ethyl-8-[4-(piperidin-3-ylmethyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
4-{4-ethoxy-3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
2,3,5-trimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-butyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-fluorophenyl)methyl]acetamide
2,2-dimethyl-4-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-3,4-dihydro-2H-pyran-6-carboxamide
3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-methyl-4-phenylpyrimidine-5-carboxamide
2-(3-phenylpropyl)-4-(thiophene-3-sulfonyl)morpholine
1-{[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-benzyl-N-methyl-3-[(4-methylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
5-({2-[4-(methylsulfamoyl)phenyl]-1H-imidazol-1-yl}methyl)thiophene-2-carboxylic acid
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-1H-pyrazole-4-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3,4-dimethylphenoxy)-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)acetamide
6-[2-(propan-2-ylsulfanyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(methylamino)pyridine-4-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidin-2-one
4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-[(4-fluorophenyl)methyl]piperazin-2-one
2-[(3-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]carbamoyl}phenyl)amino]acetic acid
2-{[(3R,4S)-4-cyclopropyl-1-(3-methoxypropanoyl)pyrrolidin-3-yl]amino}-6-(propan-2-yl)pyridine-3-carbonitrile
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthian-4-amine
N-[2-(dimethylamino)ethyl]-N,1-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-amino-4-(5-hydroxy-2-methoxyphenyl)-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide