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1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(morpholin-2-yl)ethan-1-one
2-[2-(2,3-dimethylphenoxy)ethyl]pyridin-3-ol
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-3-carboxamide
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-N-(2-chlorophenyl)propanamide
(3R,4R)-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-[2-(piperidin-2-yl)ethyl]-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-4-carboxamide
N-(3-chloro-2,6-dimethylphenyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carboxamide
3-methyl-1-[4-({3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}sulfonyl)phenyl]urea
(1S,5R)-3-[6-(4-fluorophenyl)pyridazin-3-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N3-[4-(pyridin-2-yl)pyrimidin-2-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
N-[(2-aminopyrimidin-5-yl)methyl]-3-(2-methoxyphenyl)-N-methylbenzamide
[3-(cyclopropylmethyl)-1-(4-methylpyridin-2-yl)piperidin-3-yl]methanol
{1-[1-(3,5,5-trimethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
diethyl[4-(4H-1,2,4-triazol-4-yl)pentyl]amine
(3S,4S)-4-cyclopropyl-1-(1H-imidazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
2-(2-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenoxy)acetamide
(3S,4S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-(2-methoxyethyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
3-methyl-5-{2-[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 2-[(3-{[(2-chlorophenyl)formamido]methyl}piperidine-1-carbonyl)amino]acetate
N,N-dimethyl-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}propanamide
2-(morpholin-4-yl)-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-2-(pyridin-3-yl)ethan-1-one
5-(azocane-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
1-(3-chloro-4-methoxyphenyl)-N-methyl-5-oxo-N-(pyrazin-2-ylmethyl)pyrrolidine-3-carboxamide
3-{1-[(1-benzyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}benzoic acid
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-methoxy-2-phenylethan-1-one
5-[(2S)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-ethyl-2-methyl-N-(2,2,2-trifluoroethyl)-1-benzofuran-7-carboxamide
2-methyl-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzothiazole
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-2-(2-hydroxyethyl)-3-oxo-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-6-carboxamide
3-(2-hydroxyethyl)-3-[(5-methylthiophen-2-yl)methyl]-1-[2-(propylsulfanyl)phenyl]urea
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
4-(ethylamino)-N-(2-hydroxybutyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(6-methoxypyrimidin-4-yl)amino]piperidin-1-yl}pyridine-3-carbonitrile
3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
2-ethoxy-N-methyl-N-[1-(pyridin-4-yl)ethyl]pyridine-3-carboxamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
4-(2,6-dimethylpyridin-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-2-amine
4-[1-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]morpholine
5-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
4-({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazin-2-one
diethyl({[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methyl})amine
3-(4-chloro-2,5-dimethoxyphenyl)-1-methyl-1-(oxan-2-ylmethyl)urea
5-{[4,6-dimethyl-2-(propan-2-yl)pyrimidin-5-yl]oxy}-1-azabicyclo[3.2.1]octane