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(2S)-4-methyl-N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-phenylpiperazine-1-carboxamide
N-cyclopropyl-1-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(piperidin-3-yl)benzamide
N-[(2-chlorophenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(prop-2-en-1-yl)acetamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidine-5-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-(2-ethylphenyl)-N-(3-sulfamoylphenyl)piperazine-1-carboxamide
1-(2-methoxyethyl)-5-(3-methylpiperidine-1-carbonyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
2-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)phenyl]-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-phenylpiperidine-4-carbonitrile
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,5-dimethyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-amine
(4aS,7aR)-1-[(3-chloro-4-hydroxyphenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-chlorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-cyclopropyl-4-phenyl-9-(1,3-thiazol-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2,6-dimethylpyridin-3-yl)-3-[2-(dimethylsulfamoyl)ethyl]urea
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2,4-diol
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-[2-({7-acetyl-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-4-fluorobenzamide
7-cyclohexyl-2-[(3-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4,6-dimethyl-1-(2-{4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
methyl (2S)-1-[5-(butylcarbamoyl)-1-cyclohexyl-4-oxo-1,4-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxylate
1-[(1S,5R)-6-(5-phenyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
2-{2-methyl-1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]butyl}-2,3-dihydro-1H-isoindol-1-one
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
1'-(4-chloro-2-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopropyl-1-[2-(3-methoxyphenoxy)acetyl]piperazine-2-carboxamide
N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(3-methylpyridin-4-yl)-4-[3-(methylsulfanyl)propyl]-1,4-diazepane
1-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
N-cyclopropyl-3-({1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
2-(2-butyl-1H-imidazol-4-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-3-[(4-methyl-1,4-diazepan-1-yl)methyl]benzamide
6-[(diethylamino)methyl]-N-(3-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
7-[3-(benzyloxy)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
6-methyl-5-{[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}quinoline
1-(pyridin-3-ylmethyl)-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
2-(3-chloro-4-fluorophenyl)-3-(pyrrolidine-1-carbonyl)pyridine
3-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(oxan-2-ylmethyl)benzamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]imidazolidin-2-one
N-({5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-butyl-8-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4-cycloheptylmorpholin-2-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
8-[(2R)-2-aminopropanoyl]-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one