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3-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
9-[3-(2-fluorophenyl)propanoyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidin-4-ol
5-phenyl-2-(pyridin-3-yl)-4-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]pyrimidine
8-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
4-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)benzoic acid
1-(4-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazole
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-[1-(4-acetamidobenzoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
(1R,5R)-N,N-dimethyl-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
7-amino-4-(3-hydroxy-4-methoxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1,5-dimethyl (2S)-2-{2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamido}pentanedioate
2-amino-3-ethyl-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[3-({[(9-ethyl-9H-carbazol-3-yl)methyl]amino}methyl)-5-(4-methylpiperazine-1-carbonyl)phenyl]acetamide
1-[(3-fluorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-{6-hydroxy-4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
1-cycloheptanecarbonyl-3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
1-methyl-N-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
prop-2-en-1-yl 1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carboxylate
8-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(methylsulfanyl)ethan-1-one
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-phenylpropan-1-one
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
2-(2-hydroxyethyl)-8-(3-phenylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-(3-hydroxypropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-2-carboxamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-cyclobutanecarbonyl-decahydro-1,6-naphthyridin-2-one
2-hydroxy-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
5-methyl-3-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
8-[2-(2-methoxyphenoxy)ethyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-one
(2R,3R,6R)-5-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{imidazo[1,2-a]pyridine-6-carbonyl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
methyl 2-[(2-methoxyethyl)sulfamoyl]-6-{[2-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-methoxyethyl)-9-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N3-tert-butyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2-ethoxy-5-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}phenyl)methanol
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,1,3-benzoxadiazole-5-carboxamide
2-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)-4-hydroxyquinoline-6-carboxamide
N-(2-propoxyethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidin-3-ol
1-(2-amino-6-methylpyrimidin-4-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
8-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-1-[4-(4-methyl-2-phenylpiperazine-1-carbonyl)piperidin-1-yl]ethan-1-one